SPECT imaging of glioma with radioiodinated CLINDE: evidence from a mouse GL26 glioma model
Identifieur interne : 002857 ( Main/Curation ); précédent : 002856; suivant : 002858SPECT imaging of glioma with radioiodinated CLINDE: evidence from a mouse GL26 glioma model
Auteurs : Stergios Tsartsalis [Suisse] ; Noé Dumas ; Benjamin B. Tournier ; Tien Pham ; Marcelle Moulin-Sallanon [France] ; Marie-Claude Grégoire ; Yves Charnay ; Philippe MilletSource :
- EJNMMI Research [ 2191-219X ] ; 2015.
Abstract
Recent research has demonstrated the potential of 18-kDa translocator protein (TSPO) to serve as a target for nuclear imaging of gliomas. The aim of this study was to evaluate SPECT imaging of GL26 mouse glioma using radioiodinated CLINDE, a TSPO-specific tracer.
GL26 cells, previously transfected with an enhanced green fluorescent protein (EGFP)-expressing lentivirus, were stereotactically implanted in the striatum of C57/Bl6 mice. At 4 weeks post-injection, dynamic SPECT scans with [123I]CLINDE were performed. A displacement study assessed specificity of tracer binding. SPECT images were compared to results of autoradiography, fluorescence microscopy,
Specific uptake of tracer by the tumor is observed with a high signal-to-noise ratio. Tracer uptake by the tumor is indeed 3.26 ± 0.32 times higher than that of the contralateral striatum, and 78% of the activity is displaceable by unlabeled CLINDE. Finally, TSPO is abundantly expressed by the GL26 cells.
The present study demonstrates the feasibility of [123I]CLINDE SPECT in translational studies and underlines its potential for clinical glioma SPECT imaging.
Url:
DOI: 10.1186/s13550-015-0092-4
PubMed: 25853015
PubMed Central: 4385259
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Stergios Tsartsalis<affiliation><nlm:aff id="Aff1">Vulnerability Biomarkers Unit, Division of General Psychiatry, Department of Mental Health and Psychiatry, University Hospitals of Geneva, Chemin du Petit-Bel-Air 2, CH1225 Geneva, Chêne-Bourg Switzerland</nlm:aff>
<wicri:noCountry code="subfield">Chêne-Bourg Switzerland</wicri:noCountry>
</affiliation>
<affiliation wicri:level="4"><nlm:aff id="Aff2">Department of Psychiatry, University of Geneva, 1 rue Michel-Servet, CH1211 Geneva 4, Switzerland</nlm:aff>
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<sourceDesc><biblStruct><analytic><title xml:lang="en" level="a" type="main">SPECT imaging of glioma with radioiodinated CLINDE: evidence from a mouse GL26 glioma model</title>
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<author><name sortKey="Moulin Sallanon, Marcelle" sort="Moulin Sallanon, Marcelle" uniqKey="Moulin Sallanon M" first="Marcelle" last="Moulin-Sallanon">Marcelle Moulin-Sallanon</name>
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<front><div type="abstract" xml:lang="en"><sec><title>Background</title>
<p>Recent research has demonstrated the potential of 18-kDa translocator protein (TSPO) to serve as a target for nuclear imaging of gliomas. The aim of this study was to evaluate SPECT imaging of GL26 mouse glioma using radioiodinated CLINDE, a TSPO-specific tracer.</p>
</sec>
<sec><title>Methods</title>
<p>GL26 cells, previously transfected with an enhanced green fluorescent protein (EGFP)-expressing lentivirus, were stereotactically implanted in the striatum of C57/Bl6 mice. At 4 weeks post-injection, dynamic SPECT scans with [<sup>123</sup>
I]CLINDE were performed. A displacement study assessed specificity of tracer binding. SPECT images were compared to results of autoradiography, fluorescence microscopy, <italic>in situ</italic>
nucleic acid hybridization, histology, and immunohistochemistry. Western blotting was performed to verify TSPO production by the tumor.</p>
</sec>
<sec><title>Results</title>
<p>Specific uptake of tracer by the tumor is observed with a high signal-to-noise ratio. Tracer uptake by the tumor is indeed 3.26 ± 0.32 times higher than that of the contralateral striatum, and 78% of the activity is displaceable by unlabeled CLINDE. Finally, TSPO is abundantly expressed by the GL26 cells.</p>
</sec>
<sec><title>Conclusions</title>
<p>The present study demonstrates the feasibility of [<sup>123</sup>
I]CLINDE SPECT in translational studies and underlines its potential for clinical glioma SPECT imaging.</p>
</sec>
</div>
</front>
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