Serveur d'exploration sur la rapamycine et les champignons - Exploration (Accueil)

Index « Mesh.i » - entrée « Molecular Structure »
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Molecular Sequence Data < Molecular Structure < Molecular Targeted Therapy  Facettes :

List of bibliographic references indexed by Molecular Structure

Number of relevant bibliographic references: 18.
Ident.Authors (with country if any)Title
000411 (2019) Denise Rageot [Suisse] ; Thomas Bohnacker [Suisse] ; Erhan Keles [Suisse] ; Jacob A. Mcphail [Canada] ; Reece M. Hoffmann [Canada] ; Anna Melone [Suisse] ; Chiara Borsari [Suisse] ; Rohitha Sriramaratnam [Suisse] ; Alexander M. Sele [Suisse] ; Florent Beaufils [Suisse] ; Paul Hebeisen [Suisse] ; Doriano Fabbro [Suisse] ; Petra Hillmann [Suisse] ; John E. Burke [Canada] ; Matthias P. Wymann [Suisse](S)-4-(Difluoromethyl)-5-(4-(3-methylmorpholino)-6-morpholino-1,3,5-triazin-2-yl)pyridin-2-amine (PQR530), a Potent, Orally Bioavailable, and Brain-Penetrable Dual Inhibitor of Class I PI3K and mTOR Kinase.
000483 (2018) Qingwen Huang [République populaire de Chine] ; Lijun Xie [République populaire de Chine] ; Xiaoming Chen [République populaire de Chine] ; Hui Yu [République populaire de Chine] ; Yubing Lv [République populaire de Chine] ; Xuehui Huang [République populaire de Chine] ; Jiayin Ying [République populaire de Chine] ; Congshen Zheng [République populaire de Chine] ; Yuanrong Cheng [République populaire de Chine] ; Jie Huang [République populaire de Chine]Synthesis and anticancer activity of novel rapamycin C-28 containing triazole moiety compounds.
000616 (2018) Angelina Huseinovic [Pays-Bas] ; Marc Van Dijk [Pays-Bas] ; Nico P E. Vermeulen [Pays-Bas] ; Fred Van Leeuwen [Pays-Bas] ; Jan M. Kooter [Pays-Bas] ; J Chris Vos [Pays-Bas]Drug toxicity profiling of a Saccharomyces cerevisiae deubiquitinase deletion panel shows that acetaminophen mimics tyrosine.
000632 (2018) Hairui Yang [République populaire de Chine] ; Jinsong Zhang [République populaire de Chine] ; Henan Zhang [République populaire de Chine] ; Yan Yang [République populaire de Chine] ; Yanfang Liu [République populaire de Chine] ; Wenbo Sun [République populaire de Chine] ; Wenhan Wang [République populaire de Chine] ; Wei Jia [République populaire de Chine]Compound of Stout Camphor Medicinal Mushroom, Taiwanofungus camphoratus (Agaricomycetes), Induces Protective Autophagy in SPCA-1 Cells through AMPK Inhibition-Independent Blockade of the Akt/mTOR Pathway.
000698 (2017) Hassan Y. Ebrahim [États-Unis] ; Mohamed R. Akl [États-Unis] ; Heba E. Elsayed [États-Unis] ; Ronald A. Hill [États-Unis] ; Khalid A. El Sayed [États-Unis]Usnic Acid Benzylidene Analogues as Potent Mechanistic Target of Rapamycin Inhibitors for the Control of Breast Malignancies.
000703 (2017) Eun-Hye Hong [Corée du Sud] ; Eun-Young Heo [Corée du Sud] ; Jae-Hyoung Song [Corée du Sud] ; Bo-Eun Kwon [Corée du Sud] ; Jae-Young Lee [Corée du Sud] ; Yaejeong Park [Corée du Sud] ; Jinwoong Kim [Corée du Sud] ; Sun-Young Chang [Corée du Sud] ; Young-Won Chin [Corée du Sud] ; Sang-Min Jeon [Corée du Sud] ; Hyun-Jeong Ko [Corée du Sud]Trans-scirpusin A showed antitumor effects via autophagy activation and apoptosis induction of colorectal cancer cells.
001017 (2013) Jeremy G. Owen [États-Unis] ; Boojala Vijay B. Reddy ; Melinda A. Ternei ; Zachary Charlop-Powers ; Paula Y. Calle ; Jeffrey H. Kim ; Sean F. BradyMapping gene clusters within arrayed metagenomic libraries to expand the structural diversity of biomedically relevant natural products.
001537 (2009) Flavia Marinelli [Italie]Chapter 2. From microbial products to novel drugs that target a multitude of disease indications.
001645 (2008) Jennifer L. Czlapinski [États-Unis] ; Michael W. Schelle ; Lawrence W. Miller ; Scott T. Laughlin ; Jennifer J. Kohler ; Virginia W. Cornish ; Carolyn R. BertozziConditional glycosylation in eukaryotic cells using a biocompatible chemical inducer of dimerization.
001657 (2007) R Andres Floto [Royaume-Uni] ; Sovan Sarkar ; Ethan O. Perlstein ; Beate Kampmann ; Stuart L. Schreiber ; David C. RubinszteinSmall molecule enhancers of rapamycin-induced TOR inhibition promote autophagy, reduce toxicity in Huntington's disease models and enhance killing of mycobacteria by macrophages.
001709 (2007) Michael A. Fischbach [États-Unis] ; Jon ClardyOne pathway, many products.
001848 (2005) Takuji Nakashima [Japon] ; Maki Kurachi ; Yoko Kato ; Kenichi Yamaguchi ; Tatsuya OdaCharacterization of bacterium isolated from the sediment at coastal area of Omura Bay in Japan and several biological activities of pigment produced by this isolate.
001976 (2002) R. Regentin [États-Unis] ; L. Cadapan ; S. Ou ; S. Zavala ; P. LicariProduction of a novel FK520 analog in Streptomyces hygroscopicus: improving titer while minimizing impurities.
001A10 (2001) J. Mann [Royaume-Uni]Natural products as immunosuppressive agents.
001A16 (2001) A C Gingras [Canada] ; B. Raught ; N. SonenbergControl of translation by the target of rapamycin proteins.
001A43 (2000) D A Dickman [États-Unis] ; H. Ding ; Q. Li ; A M Nilius ; D J Balli ; S J Ballaron ; J M Trevillyan ; M L Smith ; L S Seif ; K. Kim ; A. Sarthy ; R C Goldman ; J J Plattner ; Y L BennaniAntifungal rapamycin analogues with reduced immunosuppressive activity.
001A77 (1998) G K Wong [États-Unis] ; S. Griffith ; I. Kojima ; A L DemainAntifungal activities of rapamycin and its derivatives, prolylrapamycin, 32-desmethylrapamycin, and 32-desmethoxyrapamycin.
001B54 (1991) J. Heitman [Suisse] ; N R Movva ; M N HallTargets for cell cycle arrest by the immunosuppressant rapamycin in yeast.

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