Ident. | Authors (with country if any) | Title |
---|
000043 (2020) |
Fengyi Zhao [République populaire de Chine] ; Xu Sun [République populaire de Chine] ; Wen Lu [République populaire de Chine] ; Li Xu [République populaire de Chine] ; Jiuzhou Shi [République populaire de Chine] ; Shilong Yang [République populaire de Chine] ; Mengyi Zhou [République populaire de Chine] ; Fan Su [République populaire de Chine] ; Feng Lin [République populaire de Chine] ; Fuliang Cao [République populaire de Chine] | Synthesis of novel, DNA binding heterocyclic dehydroabietylamine derivatives
as potential antiproliferative and apoptosis-inducing agents |
000096 (2020) |
Ahmad Omar Noor ; Diena Mohammedallam Almasri ; Alaa Abdullah Bagalagel ; Hossam Mohamed Abdallah [Égypte] ; Shaimaa Gamal Abdallah Mohamed ; Gamal Abdallah Mohamed [Égypte] ; Sabrin Ragab Mohamed Ibrahim [Arabie saoudite, Égypte] | Naturally Occurring Isocoumarins Derivatives from Endophytic Fungi: Sources, Isolation, Structural Characterization, Biosynthesis, and Biological Activities |
000173 (2020) |
Romeol Romain Koagne [Cameroun, Espagne] ; Frederick Annang [Espagne] ; Bastien Cautain [Espagne] ; Jesús Martín [Espagne] ; Guiomar Pérez-Moreno [Espagne] ; Gabin Thierry M. Bitchagno [Cameroun] ; Dolores González-Pacanowska [Espagne] ; Francisca Vicente [Espagne] ; Ingrid Konga Simo [Cameroun] ; Fernando Reyes [Espagne] ; Pierre Tane [Cameroun] | Cytotoxycity and antiplasmodial activity of phenolic derivatives from Albizia zygia (DC.) J.F. Macbr. (Mimosaceae) |
000191 (2020) |
Wenqian Wang ; Qiuyu Meng ; Qi Li ; Jinbao Liu ; Mo Zhou [République populaire de Chine] ; Zheng Jin ; Kai Zhao [République populaire de Chine] | Chitosan Derivatives and Their Application in Biomedicine |
000224 (2020) |
Alaa Riezk [Royaume-Uni] ; John G. Raynes [Royaume-Uni] ; Vanessa Yardley [Royaume-Uni] ; Sudaxshina Murdan [Royaume-Uni] ; Simon L. Croft [Royaume-Uni] | Activity of Chitosan and Its Derivatives against Leishmania major and Leishmania mexicanaIn Vitro |
000548 (2019) |
Paolo Sgarbossa [Italie] ; Urszula Liwi Ska-Hill ; M. Fátima C. Guedes Da Silva ; Barbara Ba An W ; Aleksandra Pawlak ; Natalia Jackulak ; Dominik Poradowski ; Armando J. L. Pombeiro ; Piotr Smole Ski [Pologne] | Pentafluorophenyl Platinum(II) Complexes of PTA and Its N-Allyl and N-Benzyl Derivatives: Synthesis, Characterization and Biological Activity |
000582 (2019) |
Andrey V. Markov [Russie] ; Valeriya O. Babich [Russie] ; Irina I. Popadyuk [Russie] ; Oksana V. Salomatina [Russie] ; Evgeniya B. Logashenko [Russie] ; Nariman F. Salakhutdinov [Russie] ; Marina A. Zenkova [Russie] | Novel Derivatives of Deoxycholic Acid Bearing Linear Aliphatic Diamine and Aminoalcohol Moieties and their Cyclic Analogs at the C3 Position: Synthesis and Evaluation of Their In Vitro Antitumor Potential |
000894 (2019) |
Rui Chen [République populaire de Chine] ; Lini Huo ; Yogini Jaiswal ; Jiayong Huang ; Zhenguo Zhong ; Jing Zhong ; Leonard Williams ; Xing Xia ; Yan Liang ; Zhenshuo Yan | Design, Synthesis, Antimicrobial, and Anticancer Activities of Acridine Thiosemicarbazides Derivatives |
000921 (2019) |
Ikuko Nakamae ; Tsumoru Morimoto ; Hiroki Shima ; Masafumi Shionyu ; Hisayo Fujiki ; Noriko Yoneda-Kato ; Takashi Yokoyama ; Shigehiko Kanaya ; Kiyomi Kakiuchi ; Tsuyoshi Shirai ; Edy Meiyanto ; Jun-Ya Kato | Curcumin Derivatives Verify the Essentiality of ROS Upregulation in Tumor Suppression |
000A72 (2019) |
Branka Zorc [Croatie] ; Zrinka Raji [Croatie] ; Ivana Perkovi [Croatie] | Antiproliferative evaluation of various aminoquinoline derivatives. |
000B91 (2018-01-17) |
Jean Guillon [France] ; Anita Cohen [France] ; Rabindra Nath Das [France] ; Clotilde Boudot [France] ; Nassima Meriem Gueddouda [France] ; Stéphane Moreau [France] ; Luisa Ronga [France] ; Solène Savrimoutou [France] ; Louise Basmaciyan [France] ; Camille Tisnerat [France] ; Sacha Mestanier [France] ; Sandra Rubio [France] ; Sophia Amaziane [France] ; Alexandra Dassonville-Klimpt [France] ; Nadine Azas [France] ; Bertrand Courtioux [France] ; Jean-Louis Mergny [France] ; Catherine Mullié ; Pascal Sonnet | Design, synthesis, and antiprotozoal evaluation of new 2,9-bis[(substituted-aminomethyl)phenyl]-1,10-phenanthroline derivatives |
000B98 (2018) |
Aliasghar Jarrahpour ; Malihe Aye ; Javad Ameri Rad ; Saeed Yousefinejad [Iran] ; Veronique Sinou [France] ; Christine Latour [France] ; Jean Michel Brunel [France] ; Edward Turos | Design, synthesis, activity evaluation and QSAR studies of novel antimalarial 1,2,3-triazolo-beta-lactam derivatives |
000D34 (2016-11-26) |
J.-P. Bouillon [France] | Fluorinated mixed aminoquinoline lactam derivatives as Chloroquine-based drugs for the treatment of malaria |
000E47 (2015-05) |
Anita Cohen [France] ; Peggy Suzanne [France] ; Jean-Charles Lancelot [France] ; Pierre Verhaeghe [France] ; Aurélien Lesnard [France] ; Louise Basmaciyan [France] ; Sébastien Hutter [France] ; Michèle Laget [France] ; Aurélien Dumètre [France] ; Lucie Paloque [France] ; Eric Deharo [France] ; Maxime D. Crozet [France] ; Pascal Rathelot [France] ; Patrick Dallemagne [France] ; Audrey Lorthiois [France] ; Carol Hopkins Sibley [États-Unis] ; Patrice Vanelle [France] ; Alexis Valentin [France] ; Dominique Mazier [France] ; Sylvain Rault [France] ; Nadine Azas [France] | Discovery of new thienopyrimidinone derivatives displaying antimalarial properties toward both erythrocytic and hepatic stages of Plasmodium |
000E62 (2015) |
Patricia Melnyk [France] ; Valérie Vingtdeux [France] ; Stéphane Burlet ; Sabiha Eddarkaoui [France] ; Marie-Eve Grosjean [France] ; Paul-Emmanuel Larchanché [France] ; Guillaume Hochart [France] ; Christian Sergheraert [France] ; Cecilia Estrella ; Mathieu Barrier ; Virginie Poix ; Pauline Plancq ; Cécile Lannoo ; Malika Hamdane [France] ; André Delacourte [France] ; Philippe Verwaerde ; Luc Buee [France] ; Nicolas Sergeant [France] | Chloroquine and Chloroquinoline Derivatives as Models for the Design of Modulators of Amyloid Peptide Precursor Metabolism |
000F90 (2014-12-03) |
Maribel Navarro [Venezuela] ; William Castro [Venezuela] ; Marilyn Madamet [France] ; Rémy Amalvict [France] ; Nicolas Benoit [France] ; Bruno Pradines [France] | Metal-chloroquine derivatives as possible anti-malarial drugs: evaluation of anti-malarial activity and mode of action |
001000 (2014) |
Issaka Sagara [Mali] ; Renaud Piarroux [France] ; Abdoulaye Djimde [Mali] ; Roch Giorgi [France] ; Kassoum Kayentao [Mali] ; Ogobara Doumbo [Mali] ; Jean Gaudart [France] | Delayed anemia assessment in patients treated with oral artemisinin derivatives for uncomplicated malaria: a pooled analysis of clinical trials data from Mali. |
001023 (2014) |
Jennifer Keiser [Suisse] ; Mireille Vargas ; Riccardo Rubbiani ; Gilles Gasser ; Christophe Biot | In vitro and in vivo antischistosomal activity of ferroquine derivatives. |
001037 (2014) |
Andreia Montoia [Brésil] ; Luiz F. Rocha E Silva [Brésil] ; Zelina E. Torres [Brésil] ; David S. Costa [Brésil] ; Marycleuma C. Henrique [Brésil] ; Emerson S. Lima [Brésil] ; Marne C. Vasconcellos [Brésil] ; Rita C Z. Souza [Brésil] ; Monica R F. Costa [Brésil] ; Andriy Grafov [Finlande] ; Iryna Grafova [Finlande] ; Marcos N. Eberlin [Brésil] ; Wanderli P. Tadei [Brésil] ; Rodrigo C N. Amorim [Brésil] ; Adrian M. Pohlit [Brésil] | Antiplasmodial activity of synthetic ellipticine derivatives and an isolated analog. |
001159 (2013) |
Weijie Li [République populaire de Chine] ; Jing Hao [République populaire de Chine] ; Yeyu Xiao [République populaire de Chine] | Synthesis and in vitro antitumor activities of lupeol dicarboxylic acid monoester derivatives |
001276 (2012-08) |
Luke Mani ; Valerie Jullian ; Beatrice Mourkazel ; Alexis Valentin ; Joëlle Dubois [France] ; Thierry Cresteil [France] ; Eric Folcher ; John N A. Hooper ; Dirk Erpenbeck ; William Aalbersberg ; Cécile Debitus | New antiplasmodial bromotyrosine derivatives from Suberea ianthelliformis Lendenfeld, 1888. |