001A39 (2008) |
Sandrine Delarue-Cochin [France] ; Philippe Grellier [France] ; Louis Maes [Belgique] ; Elisabeth Mouray [France] ; Christian Sergheraert [France] ; Patricia Melnyk [France] | Synthesis and antimalarial activity of carbamate and amide derivatives of 4-anilinoquinoline |
002040 (2003) |
Adina Ryckebusch [Belgique] ; Rébecca Deprez-Poulain [Belgique] ; Louis Maes [Belgique] ; Marie-Ange Debreu-Fontaine [Belgique] ; Elisabeth Mouray [Belgique] ; Philippe Grellier [Belgique] ; Christian Sergheraert [Belgique, France] | Synthesis and in Vitro and in Vivo Antimalarial Activity of N-(7-Chloro-4-quinolyl)-1,4-bis(3-aminopropyl)piperazine Derivatives |
002285 (2001) |
Sophie Girault [Belgique] ; Philippe Grellier [Belgique] ; Amaya Berecibar [Belgique, France] ; Louis Maes [Belgique] ; Pascal Lemière [Belgique] ; Elisabeth Mouray [Belgique] ; Elisabeth Davioud-Charvet [Belgique] ; Christian Sergheraert [Belgique, France] | Antiplasmodial Activity and Cytotoxicity of Bis-, Tris-, and Tetraquinolines with Linear or Cyclic Amino Linkers |
002471 (2000) |
Sophie Girault [Belgique] ; Philippe Grellier [Belgique] ; Amaya Berecibar [Belgique] ; Louis Maes [Belgique] ; Elisabeth Mouray [Belgique] ; Pascal Lemière [Belgique] ; Marie-Ange Debreu [Belgique] ; Elisabeth Davioud-Charvet [Belgique] ; Christian Sergheraert [Belgique, France] | Antimalarial, Antitrypanosomal, and Antileishmanial Activities and Cytotoxicity of Bis(9-amino-6-chloro-2-methoxyacridines): Influence of the Linker# |
000739 (2019) |
R Kanyanga Cimanga [Belgique] ; S Lumpu Nsaka ; M Ehata Tshodi ; B Maya Mbamu ; C Munduku Kikweta ; F Bool-Miting Makila ; Paul Cos [Belgique] ; Louis Maes [Belgique] ; Arnold J. Vlietinck [Belgique] ; Vassiliki Exarchou [Belgique] ; Emmy Tuenter [Belgique] ; Luc Pieters [Belgique] | In vitro and in vivo antiplasmodial activity of extracts and isolated constituents of Alstonia congensis root bark. |
000785 (2019) |
Yancho Zarev [Belgique] ; Kenn Foubert [Belgique] ; Paul Cos [Belgique] ; Louis Maes [Belgique] ; Esameldin Elgorashi [Afrique du Sud] ; Sandra Apers [Belgique] ; Iliana Ionkova [Bulgarie] ; Luc Pieters [Belgique] | HPLC-DAD-SPE-NMR isolation of tetracyclic spiro-alkaloids with antiplasmodial activity from the seeds of Erythrina latissima. |
001404 (2012) |
Mehdi A. Beniddir ; Philippe Grellier [France] ; Philippe Rasoanaivo [Madagascar] ; Philippe M. Loiseau [France] ; Christian Bories [France] ; Vincent Dumontet ; Françoise Guéritte ; Marc Litaudon [France] | Diarylheptanoid Glucosides from Pyrostria major and Their Antiprotozoal Activities |
001604 (2010-10) |
Mélanie Bourjot ; Cécile Apel [France] ; Marie-Thérèse Martin [France] ; Philippe Grellier ; Van Hung Nguyen [France] ; Françoise Guéritte [France] ; Marc Litaudon [France] | Antiplasmodial, antitrypanosomal, and cytotoxic activities of prenylated flavonoids isolated from the stem bark of Artocarpus styracifolius. |
001606 (2010-06) |
Guillaume Marti [France] ; Véronique Eparvier [France] ; Christian Moretti ; Soizic Prado ; Philippe Grellier ; Nathalie Hue ; Odile Thoison [France] ; Bernard Delpech [France] ; Françoise Guéritte [France] ; Marc Litaudon [France] | Antiplasmodial benzophenone derivatives from the root barks of Symphonia globulifera (Clusiaceae). |
001625 (2010) |
Kahunu Mesia ; Richard K. Cimanga ; Liene Dhooghe ; Paul Cos ; Sandra Apers ; Jozef Totté ; Gaston L. Tona ; Luc Pieters ; Arnold J. Vlietinck ; Louis Maes | Antimalarial activity and toxicity evaluation of a quantified Nauclea pobeguinii extract. |
001628 (2010) |
Guillaume Marti [France] ; Véronique Eparvier ; Marc Litaudon ; Philippe Grellier ; Françoise Guéritte | A new xanthone from the bark extract of Rheedia acuminata and antiplasmodial activity of its major compounds. |
001763 (2010) |
Kahunu Mesia [République du Congo, Belgique] ; Richard K. Cimanga [République du Congo, Belgique] ; Liene Dhooghe [Belgique] ; Paul Cos [Belgique] ; Sandra Apers [Belgique] ; Jozef Totte [Belgique] ; Gaston L. Tona [République du Congo] ; Luc Pieters [Belgique] ; Arnold J. Vlietinck [Belgique] ; Louis Maes [Belgique] | Antimalarial activity and toxicity evaluation of a quantified Nauclea pobeguinii extract |
001774 (2009-01) |
Guillaume Marti [France] ; Véronique Eparvier [France] ; Christian Moretti [France] ; Sophie Susplugas ; Soizic Prado [France] ; Philippe Grellier [France] ; Pascal Retailleau [France] ; Françoise Guéritte [France] ; Marc Litaudon [France] | Antiplasmodial benzophenones from the trunk latex of Moronobea coccinea (Clusiaceae). |
002260 (2001) |
Sandrine Delarue [Belgique] ; Sophie Girault [Belgique] ; Louis Maes [Belgique] ; Marie-Ange Debreu-Fontaine [Belgique] ; Mehdi Labaeïd [Belgique] ; Philippe Grellier [Belgique] ; Christian Sergheraert [Belgique, France] | Synthesis and in Vitro and in Vivo Antimalarial Activity of New 4-Anilinoquinolines† |
002289 (2001) |
Elisabeth Davioud-Charvet [Allemagne, États-Unis] ; Sandrine Delarue [Allemagne] ; Christophe Biot [Allemagne] ; Babett Schwöbel [Allemagne] ; Catharina C. Boehme [Allemagne] ; Andreas Müssigbrodt [Allemagne] ; Louis Maes [Allemagne] ; Christian Sergheraert [Allemagne] ; Philippe Grellier [Allemagne] ; R. Heiner Schirmer [Allemagne] ; Katja Becker [Allemagne] | A Prodrug Form of a Plasmodium falciparum Glutathione Reductase Inhibitor Conjugated with a 4-Anilinoquinoline |
000F81 (2015) |
Osmany Cuesta-Rubio [Équateur] ; Ahmad Oubada [Cuba] ; Adonis Bello [Équateur] ; Louis Maes [Belgique] ; Paul Cos [Belgique] ; Lianet Monzote [Cuba] | Antimicrobial Assessment of Resins from Calophyllum Antillanum and Calophyllum Inophyllum |
001062 (2014) |
Soraia I. Falcão [Portugal] ; Nuno Vale [Portugal] ; Paul Cos [Belgique] ; Paula Gomes [Portugal] ; Cristina Freire [Portugal] ; Louis Maes [Belgique] ; Miguel Vilas-Boas [Portugal] | In Vitro Evaluation of Portuguese Propolis and Floral Sources for Antiprotozoal, Antibacterial and Antifungal Activity |
001463 (2011) |
Kevin Spelman [États-Unis] ; Delphine Depoix [France] ; Megan Mccray [États-Unis] ; Elisabeth Mouray [France] ; Philippe Grellier [France] | The Traditional Medicine Spilanthes acmella, and the Alkylamides Spilanthol and Undeca-2E-ene-8,10-diynoic Acid Isobutylamide, Demonstrate In Vitro and In Vivo Antimalarial Activity |
001464 (2011) |
Pieter Leyssen [Belgique] ; Marc Litaudon [France] ; Jean-Claude Guillemot [France] ; Philippe Rasoanaivo [Madagascar] ; Jacqueline Smadja [Réunion] ; Ameenah Gurib-Fakim ; Bruno Canard [France] ; Françoise Guéritte [France] | PHYTOCHIK: Biodiversity As A Source of Selective Inhibitors of CHIKV Replication |
001824 (2009) |
Emilia P Unescu [Roumanie] ; Sophie Susplugas [France] ; Emmanuelle Boll ; Richard Varga [Roumanie] ; Elisabeth Mouray [France] ; Ion Grosu [Roumanie] ; Philippe Grellier [France] ; Patricia Melnyk [France] | Replacement of the 4′‐Hydroxy Group of Amodiaquine and Amopyroquine by Aromatic and Aliphatic Substituents: Synthesis and Antimalarial Activity |
001927 (2008) |
E. Paunescu [France] ; Sophie Susplugas [France] ; E. Boll ; R. Varga ; Elisabeth Mouray [France] ; Philippe Grellier [France] ; Patricia Melnyk [France] | Synthesis and antimalarial activity of new amino analogues of amodiaquine. |
001A43 (2008) |
Voahangy Ramanandraibe [Madagascar] ; Philippe Grellier [France] ; Marie-Thérèse Martin [France] ; Alexandre Deville [France] ; Roger Joyeau [France] ; David Ramanitrahasimbola [Madagascar] ; Elisabeth Mouray [France] ; Philippe Rasoanaivo [Madagascar] ; Lengo Mambu [France] | Antiplasmodial Phenolic Compounds from Piptadenia pervillei |
001C10 (2006) |
Patricia Melnyk [France] ; Virginie Leroux [France] ; Christian Sergheraert [France] ; Philippe Grellier [France] | Design, synthesis and in vitro antimalarial activity of an acylhydrazone library |
002162 (2002) |
Tim H. M. Jonckers [Belgique] ; Sabine Van Miert [Belgique] ; Kanyanga Cimanga [Belgique] ; Christian Bailly [Belgique] ; Pierre Colson [Belgique] ; Marie-Claire De Pauw-Gillet [Belgique] ; Hilde Van Den Heuvel [Belgique] ; Magda Claeys [Belgique] ; Filip Lemière [Belgique] ; Eddy L. Esmans [Belgique] ; Jef Rozenski [Belgique] ; Ludo Quirijnen [Belgique] ; Louis Maes [Belgique] ; Roger Dommisse [Belgique] ; Guy L. F. Lemière [Belgique] ; Arnold Vlietinck [Belgique] ; Luc Pieters [Belgique] | Synthesis, Cytotoxicity, and Antiplasmodial and Antitrypanosomal Activity of New Neocryptolepine Derivatives |
000E23 (2016) |
Yamilet Gutiérrez [Cuba] ; Rodny Montes [Cuba] ; Ram N Scull [Cuba] ; Arturo Sánchez [Cuba] ; Paul Cos ; Lianet Monzote [Cuba] ; William N. Setzer [États-Unis] | Chemodiversity Associated with Cytotoxicity and Antimicrobial Activity of Piper aduncum var. ossanum |
000E62 (2015) |
Patricia Melnyk [France] ; Valérie Vingtdeux [France] ; Stéphane Burlet ; Sabiha Eddarkaoui [France] ; Marie-Eve Grosjean [France] ; Paul-Emmanuel Larchanché [France] ; Guillaume Hochart [France] ; Christian Sergheraert [France] ; Cecilia Estrella ; Mathieu Barrier ; Virginie Poix ; Pauline Plancq ; Cécile Lannoo ; Malika Hamdane [France] ; André Delacourte [France] ; Philippe Verwaerde ; Luc Buee [France] ; Nicolas Sergeant [France] | Chloroquine and Chloroquinoline Derivatives as Models for the Design of Modulators of Amyloid Peptide Precursor Metabolism |
001027 (2014) |
Jane Namukobe [Ouganda] ; Bernard T. Kiremire [Ouganda] ; Robert Byamukama [Ouganda] ; John M. Kasenene [Ouganda] ; Vincent Dumontet [France] ; Françoise Guéritte [France] ; Sabrina Krief [Ouganda] ; Isabelle Florent [France] ; John D. Kabasa [Ouganda] | Cycloartane triterpenes from the leaves of Neoboutonia macrocalyx L. |
001093 (2013-07-22) |
Faustine Dubar [France] ; Christian Slomianny [France] ; Jamal Khalife [France] ; Daniel Dive [France] ; Hadidjatou Kalamou [France] ; Yann Guerardel [France] ; Philippe Grellier [France] ; Christophe Biot [France] | The Ferroquine Antimalarial Conundrum: Redox Activation and Reinvasion Inhibition |
001126 (2013) |
Fereshteh Farokhi [France] ; Philippe Grellier ; Monique Clément ; Christos Roussakis ; Philippe M. Loiseau ; Emilie Genin-Seward ; Jean-Michel Kornprobst ; Gilles Barnathan ; Gaëtane Wielgosz-Collin | Antimalarial activity of axidjiferosides, new β-galactosylceramides from the African sponge Axinyssa djiferi. |
001654 (2010) |
Claire Madelaine [France] ; Olivier Buriez [France] ; Benot Crousse [France] ; Isabelle Florent [France] ; Philippe Grellier [France] ; Pascal Retailleau [France] ; Yvan Six [France] | Aminocyclopropanes as precursors of endoperoxides with antimalarial activity |
001713 (2010) |
Gesine Bradacs [Allemagne] ; Louis Maes [Belgique] ; Jörg Heilmann [Allemagne] | In vitro cytotoxic, antiprotozoal and antimicrobial activities of medicinal plants from Vanuatu |
001714 (2010) |
Essam Abdel-Sattar [Arabie saoudite] ; Louis Maes [Belgique] ; Maha Mahmoud Salama [Égypte] | In Vitro activities of plant extracts from Saudi Arabia against malaria, leishmaniasis, sleeping sickness and Chagas disease |
001745 (2010) |
Jean Gustave Tangmouo [Cameroun, Suisse] ; Raimana Ho [Suisse] ; An Matheeussen [Belgique] ; Alain Meli Lannang [Cameroun] ; Justin Komguem [Cameroun] ; Bernadette Biloa Messi [Cameroun, Suisse] ; Louis Maes [Belgique] ; Kurt Hostettmann [Suisse] | Antimalarial activity of extract and norbergenin derivatives from the stem bark of Diospyros sanza‐minika A. Chevalier (Ebenaceae) |
001A59 (2007) |
Julie Nguyen-Pouplin [France] ; Hop Tran ; Hung Tran ; Tuyet Anh Phan ; Christiane Dolecek ; Jeremy Farrar ; Tinh Hien Tran ; Philippe Caron ; Bernard Bodo ; Philippe Grellier | Antimalarial and cytotoxic activities of ethnopharmacologically selected medicinal plants from South Vietnam. |
001E02 (2005-05-16) |
Guédé Noël Zirihi ; Philippe Grellier [France] ; Frédérick Guédé-Guina ; Bernard Bodo [France] ; Lengo Mambu [France] | Isolation, characterization and antiplasmodial activity of steroidal alkaloids from Funtumia elastica (Preuss) Stapf. |
002C34 (1994) |
Frédérick Gay [France] ; Liliane Ciceron [France] ; Marc Litaudon [France] ; Madorina Bustos [France] ; Pascal Astagneau [France] ; Bertrand Diquet [France] ; Martin Danis [France] ; Marc Gentilini [France] | In-vitro resistance of Plasmodium falciparum to qinghaosu derivatives in West Africa |
003037 (1990) |
Frédérick Gay [France] ; Dorinag. Bustos [France] ; Bertrand Diquet [France] ; Lazara Rojas Rivero [France] ; Marc Litaudon [France] ; Christian Pichet [France] ; Martin Danis [France] ; Marc Gentilini [France] | Cross-resistance between mefloquine and halofantrine |