List of bibliographic references
Number of relevant bibliographic references: 15.
Ident. | Authors (with country if any) | Title |
---|
000241 (2019) |
Denise Rageot [Suisse] ; Thomas Bohnacker [Suisse] ; Erhan Keles [Suisse] ; Jacob A. Mcphail [Canada] ; Reece M. Hoffmann [Canada] ; Anna Melone [Suisse] ; Chiara Borsari [Suisse] ; Rohitha Sriramaratnam [Suisse] ; Alexander M. Sele [Suisse] ; Florent Beaufils [Suisse] ; Paul Hebeisen [Suisse] ; Doriano Fabbro [Suisse] ; Petra Hillmann [Suisse] ; John E. Burke [Canada] ; Matthias P. Wymann [Suisse] | (S)-4-(Difluoromethyl)-5-(4-(3-methylmorpholino)-6-morpholino-1,3,5-triazin-2-yl)pyridin-2-amine (PQR530), a Potent, Orally Bioavailable, and Brain-Penetrable Dual Inhibitor of Class I PI3K and mTOR Kinase. |
000309 (2019) |
Patrick Schwarz [Allemagne] ; Petra V. Schwarz [Allemagne] ; Heike Felske-Zech [Allemagne] ; Eric Dannaoui [France] | In vitro interactions between isavuconazole and tacrolimus, cyclosporin A or sirolimus against Mucorales. |
000314 (2019) |
Yueh-Han Hsu [Taïwan] ; Hui-Pei Huang [Taïwan] ; Horng-Rong Chang [Taïwan] | The uremic toxin p-cresol promotes the invasion and migration on carcinoma cells via Ras and mTOR signaling. |
000420 (2018) |
Denise Rageot [Suisse] ; Thomas Bohnacker [Suisse] ; Anna Melone [Suisse] ; Jean-Baptiste Langlois [Suisse] ; Chiara Borsari [Suisse] ; Petra Hillmann [Suisse] ; Alexander M. Sele [Suisse] ; Florent Beaufils [Suisse] ; Marketa Zvelebil [Suisse] ; Paul Hebeisen [Suisse] ; Wolfgang Löscher [Allemagne] ; John Burke [Canada] ; Doriano Fabbro [Suisse] ; Matthias P. Wymann [Suisse] | Discovery and Preclinical Characterization of 5-[4,6-Bis({3-oxa-8-azabicyclo[3.2.1]octan-8-yl})-1,3,5-triazin-2-yl]-4-(difluoromethyl)pyridin-2-amine (PQR620), a Highly Potent and Selective mTORC1/2 Inhibitor for Cancer and Neurological Disorders. |
000513 (2018) |
Angela Kwok-Fung Lo [Hong Kong] ; Raymond Wai-Ming Lung [Hong Kong] ; Christopher W. Dawson [Royaume-Uni] ; Lawrence S. Young [Royaume-Uni] ; Chuen-Wai Ko [Hong Kong] ; Walter Wai Yeung [Hong Kong] ; Wei Kang [Hong Kong] ; Ka-Fai To [Hong Kong] ; Kwok-Wai Lo [Hong Kong] | Activation of sterol regulatory element-binding protein 1 (SREBP1)-mediated lipogenesis by the Epstein-Barr virus-encoded latent membrane protein 1 (LMP1) promotes cell proliferation and progression of nasopharyngeal carcinoma. |
000582 (2018) |
Chunhui Wang [République populaire de Chine] ; Jianghong Qu [République populaire de Chine] ; Siyuan Yan [République populaire de Chine] ; Quan Gao [République populaire de Chine] ; Sibin Hao [République populaire de Chine] ; Dongsheng Zhou [République populaire de Chine] | PFK15, a PFKFB3 antagonist, inhibits autophagy and proliferation in rhabdomyosarcoma cells. |
000749 (2017) |
Inan Olmez [États-Unis] ; Breanna Brenneman [États-Unis] ; Aizhen Xiao [États-Unis] ; Vlad Serbulea [États-Unis] ; Mouadh Benamar [États-Unis] ; Ying Zhang [États-Unis] ; Laryssa Manigat [États-Unis] ; Tarek Abbas [États-Unis] ; Jeongwu Lee [États-Unis] ; Ichiro Nakano [États-Unis] ; Jakub Godlewski [États-Unis] ; Agnieszka Bronisz [États-Unis] ; Roger Abounader [États-Unis] ; Norbert Leitinger [États-Unis] ; Benjamin Purow [États-Unis] | Combined CDK4/6 and mTOR Inhibition Is Synergistic against Glioblastoma via Multiple Mechanisms. |
000812 (2017) |
Kwang-Youn Kim [Corée du Sud] ; Kwang-Il Park [Corée du Sud] ; Sang-Hun Kim [Corée du Sud] ; Sun-Nyoung Yu [Corée du Sud] ; Sul-Gi Park [Corée du Sud] ; Young Woo Kim [Corée du Sud] ; Young-Kyo Seo [Corée du Sud] ; Jin-Yeul Ma [Corée du Sud] ; Soon-Cheol Ahn [Corée du Sud] | Inhibition of Autophagy Promotes Salinomycin-Induced Apoptosis via Reactive Oxygen Species-Mediated PI3K/AKT/mTOR and ERK/p38 MAPK-Dependent Signaling in Human Prostate Cancer Cells. |
000A28 (2016) |
Yan Sun [États-Unis] ; Jonathan O. Lipton [États-Unis] ; Lara M. Boyle [États-Unis] ; Joseph R. Madsen [États-Unis] ; Marti C. Goldenberg [États-Unis] ; Alvaro Pascual-Leone [États-Unis] ; Mustafa Sahin [États-Unis] ; Alexander Rotenberg [États-Unis] | Direct current stimulation induces mGluR5-dependent neocortical plasticity. |
000F51 (2013) |
Dae Won Park [Corée du Sud] ; Shaoning Jiang [États-Unis] ; Jean-Marc Tadie [France] ; William S. Stigler [États-Unis] ; Yong Gao [États-Unis] ; Jessy Deshane [États-Unis] ; Edward Abraham [États-Unis] ; Jaroslaw W. Zmijewski [États-Unis] | Activation of AMPK enhances neutrophil chemotaxis and bacterial killing. |
000F81 (2014) |
Tiffany N. Caza [États-Unis] ; David R. Fernandez [États-Unis] ; Gergely Talaber [États-Unis] ; Zachary Oaks [États-Unis] ; Mark Haas [États-Unis] ; Michael P. Madaio [États-Unis] ; Zhi-Wei Lai [États-Unis] ; Gabriella Miklossy [États-Unis] ; Ram R. Singh [États-Unis] ; Dmitriy M. Chudakov [Russie] ; Walter Malorni [Italie] ; Frank Middleton [États-Unis] ; Katalin Banki [États-Unis] ; Andras Perl [États-Unis] | HRES-1/Rab4-mediated depletion of Drp1 impairs mitochondrial homeostasis and represents a target for treatment in SLE. |
001271 (2012) |
Fabrizio Di Benedetto ; Massimiliano Berretta ; Nicola De Ruvo ; Giuseppe Tarantino ; Giuseppe D'Amico ; Roberto Ballarin ; Rosa Maria Iemmolo ; Giorgio E. Gerunda | Is advanced hepatocellular carcinoma amenable of cure by liver transplantation with sorafenib as a neoadjuvant approach plus m-TOR inhibitors monotherapy? |
001629 (2008) |
H Reynaldo L Pez-Mirabal [Danemark] ; Jakob R. Winther ; Morten C. Kielland-Brandt | Oxidant resistance in a yeast mutant deficient in the Sit4 phosphatase. |
001857 (2004) |
Mercedes B. Fuertes [Argentine] ; Luciana L. Molinero ; Marta A. Toscano ; Juan M. Ilarregui ; Natalia Rubinstein ; Leonardo Fainboim ; Norberto W. Zwirner ; Gabriel A. Rabinovich | Regulated expression of galectin-1 during T-cell activation involves Lck and Fyn kinases and signaling through MEK1/ERK, p38 MAP kinase and p70S6 kinase. |
001A22 (2001) |
A. Gagnon [Canada] ; P. Dods ; N. Roustan-Delatour ; C S Chen ; A. Sorisky | Phosphatidylinositol-3,4,5-trisphosphate is required for insulin-like growth factor 1-mediated survival of 3T3-L1 preadipocytes. |
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