Serveur d'exploration SRAS

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Inhibiteur reverse transcriptase And NotFen-Er Chen

List of bibliographic references

Number of relevant bibliographic references: 7.
Ident.Authors (with country if any)Title
000198 Andrea Spallarossa [Italie] ; Sara Cesarini [Italie] ; Angelo Ranise [Italie] ; Silvia Schenone [Italie] ; Olga Bruno [Italie] ; Alberto Borassi [Italie] ; Paolo La Colla [Italie] ; Margherita Pezzullo [Italie] ; Giuseppina Sanna [Italie] ; Gabriella Collu [Italie] ; Barbara Secci [Italie] ; Roberta Loddo [Italie]Parallel synthesis, molecular modelling and further structure-activity relationship studies of new acylthiocarbamates as potent non-nucleoside HIV-1 reverse transcriptase inhibitors
000200 Andrea Spallarossa [Italie] ; Sara Cesarini [Italie] ; Angelo Ranise [Italie] ; Olga Bruno [Italie] ; Silvia Schenone [Italie] ; Paolo La Colla [Italie] ; Gabriella Collu [Italie] ; Giuseppina Sanna [Italie] ; Barbara Secci [Italie] ; Roberta Loddo [Italie]Novel modifications in the series of O-(2-phthalimidoethyl)-N-substituted thiocarbamates and their ring-opened congeners as non-nucleoside HIV-1 reverse transcriptase inhibitors
000237 Sara Cesarini [Italie] ; Andrea Spallarossa [Italie] ; Angelo Ranise [Italie] ; Olga Bruno [Italie] ; Paolo La Colla [Italie] ; Barbara Secci [Italie] ; Gabriella Collu [Italie] ; Roberta Loddo [Italie]Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 2. Parallel synthesis, molecular modelling and structure-activity relationship studies on analogues of O-(2-phenylethyl)-N-phenylthiocarbamate
000238 Sara Cesarini [Italie] ; Andrea Spallarossa [Italie] ; Angelo Ranise [Italie] ; Paola Fossa [Italie] ; Paolo La Colla [Italie] ; Giuseppina Sanna [Italie] ; Gabriella Collu [Italie] ; Roberta Loddo [Italie]Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 1. Parallel synthesis, molecular modelling and structure-activity relationship studies on 0-[2-(hetero)arylethyl]-N-phenylthiocarbamates
000565 Naoyuki Masuda [Japon] ; Osamu Yamamoto [Japon] ; Masahiro Fujii [Japon] ; Tetsuro Ohgami [Japon] ; Jiro Fujiyasu [Japon] ; Toru Kontani [Japon] ; Ayako Moritomo [Japon] ; Masaya Orita [Japon] ; Hiroyuki Kurihara [Japon] ; Hironobu Koga [Japon] ; Shunji Kageyama [Japon] ; Mitsuaki Ohta [Japon] ; Hiroshi Inoue [Japon] ; Toshifumi Hatta [Japon] ; Masafumi Shintani [Japon] ; Hiroshi Suzuki [Japon] ; Kenji Sudo [Japon] ; Yasuaki Shimizu [Japon] ; Eiichi Kodama [Japon] ; Masao Matsuoka [Japon] ; Masatoshi Fujiwara [Japon] ; Tomoyuki Yokota [Japon] ; Shiro Shigeta [Japon] ; Masanori Baba [Japon]Studies of non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 2: Synthesis and structure-activity relationships of 2-cyano and 2-hydroxy thiazolidenebenzenesulfonamide derivatives
000571 Caterina Fattorusso [Italie] ; Sandra Gemma [Italie] ; Stefania Butini [Italie] ; Paul Huleatt [Italie] ; Bruno Catalanotti [Italie] ; Marco Persico [Italie] ; Meri De Angelis [Italie] ; Isabella Fiorini [Italie] ; V Ito Nacci [Italie] ; Anna Ramunno [Italie] ; Manuela Rodriquez [Italie] ; Giovanni Greco [Italie] ; Ettore Novellino [Italie] ; Alberto Bergamini [Italie] ; Stefano Marini [Italie] ; Massimo Coletta [Italie] ; Giovanni Maga [Italie] ; Silvio Spadari [Italie] ; Giuseppe Campiani [Italie]Specific targeting highly conserved residues in the HIV-1 reverse transcriptase primer grip region. design, synthesis, and biological evaluation of novel, potent, and broad spectrum NNRTIs with antiviral activity
000972 Angelo Ranise [Italie] ; Andrea Spallarossa [Italie] ; Silvia Schenone [Italie] ; Olga Bruno [Italie] ; Francesco Bondavalli [Italie] ; Laura Vargiu [Italie] ; Tiziana Marceddu [Italie] ; Massimo Mura [Italie] ; Paolo La Colla [Italie] ; Alessandra Pani [Italie]Design, synthesis, SAR, and molecular modeling studies of acylthiocarbamates: A novel series of potent non-nucleoside HIV-1 reverse transcriptase inhibitors structurally related to phenethylthiazolylthiourea derivatives

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