| Ident. | Authors (with country if any) | Title |
|---|
| 001563 (2006) |
Hui Li [États-Unis] ; John Tatlock ; Angelica Linton ; Javier Gonzalez ; Allen Borchardt ; Peter Dragovich ; Tanya Jewell ; Tom Prins ; Ru Zhou ; Julie Blazel ; Hans Parge ; Robert Love ; Michael Hickey ; Chau Doan ; Stephanie Shi ; Rohit Duggal ; Cristina Lewis ; Shella Fuhrman | Identification and structure-based optimization of novel dihydropyrones as potent HCV RNA polymerase inhibitors. |
| 001593 (2006) |
Yue-Qing Li [République populaire de Chine] ; Ze-Lin Li ; Wei-Jie Zhao ; Rui-Xing Wen ; Qing-Wei Meng ; Yi Zeng | Synthesis of stilbene derivatives with inhibition of SARS coronavirus replication. |
| 001599 (2006) |
Syaulan Yang [République populaire de Chine] ; Shu-Jen Chen ; Min-Feng Hsu ; Jen-Dar Wu ; Chien-Te K. Tseng ; Yu-Fan Liu ; Hua-Chien Chen ; Chun-Wei Kuo ; Chi-Shen Wu ; Li-Wen Chang ; Wen-Chang Chen ; Shao-Ying Liao ; Teng-Yuan Chang ; Hsin-Hui Hung ; Hui-Lin Shr ; Cheng-Yuan Liu ; Yu-An Huang ; Ling-Yin Chang ; Jen-Chi Hsu ; Clarence J. Peters ; Andrew H-J Wang ; Ming-Chu Hsu | Synthesis, crystal structure, structure-activity relationships, and antiviral activity of a potent SARS coronavirus 3CL protease inhibitor. |
| 001614 (2006) |
Pamela Hamill [Canada] ; Derek Hudson ; Richard Y. Kao ; Polly Chow ; Meera Raj ; Hongyan Xu ; Martin J. Richer ; François Jean | Development of a red-shifted fluorescence-based assay for SARS-coronavirus 3CL protease: identification of a novel class of anti-SARS agents from the tropical marine sponge Axinella corrugata. |
| 001623 (2006) |
I-Lin Lu [République populaire de Chine] ; Neeraj Mahindroo ; Po-Huang Liang ; Yi-Hui Peng ; Chih-Jung Kuo ; Keng-Chang Tsai ; Hsing-Pang Hsieh ; Yu-Sheng Chao ; Su-Ying Wu | Structure-based drug design and structural biology study of novel nonpeptide inhibitors of severe acute respiratory syndrome coronavirus main protease. |
| 001669 (2007) |
S-Q Wang [République populaire de Chine] ; Q-S Du ; K. Zhao ; A-X Li ; D-Q Wei ; K-C Chou | Virtual screening for finding natural inhibitor against cathepsin-L for SARS therapy. |
| 001726 (2006) |
Rolf Hilgenfeld [Allemagne] ; Kanchan Anand ; Jeroen R. Mesters ; Zihe Rao ; Xu Shen ; Hualiang Jiang ; Jinzhi Tan ; Koen H G. Verschueren | Structure and dynamics of SARS coronavirus main proteinase (Mpro). |
| 001737 (2006) |
Lili Chen [République populaire de Chine] ; Jian Li ; Cheng Luo ; Hong Liu ; Weijun Xu ; Gang Chen ; Oi Wah Liew ; Weiliang Zhu ; Chum Mok Puah ; Xu Shen ; Hualiang Jiang | Binding interaction of quercetin-3-beta-galactoside and its synthetic derivatives with SARS-CoV 3CL(pro): structure-activity relationship studies reveal salient pharmacophore features. |
| 001761 (2006) |
Lili Chen [République populaire de Chine] ; Shuai Chen ; Chunshan Gui ; Jianhua Shen ; Xu Shen ; Hualiang Jiang | Discovering severe acute respiratory syndrome coronavirus 3CL protease inhibitors: virtual screening, surface plasmon resonance, and fluorescence resonance energy transfer assays. |
| 001805 (2006) |
Haitao Yang [République populaire de Chine] ; Mark Bartlam ; Zihe Rao | Drug design targeting the main protease, the Achilles' heel of coronaviruses. |
| 001809 (2006) |
Chung K. Chu [États-Unis] ; Srinivas Gadthula ; Xin Chen ; Hyunah Choo ; Sureyya Olgen ; Dale L. Barnard ; Robert W. Sidwell | Antiviral activity of nucleoside analogues against SARS-coronavirus (SARS-coV). |
| 001901 (????) |
Q-Y Yang [République populaire de Chine] ; X-Y Tian ; W-S Fang | Bioactive coumarins from Boenninghausenia sessilicarpa. |
| 001B02 (2007) |
Cheng-Chung Lee [Taïwan] ; Chih-Jung Kuo ; Min-Feng Hsu ; Po-Huang Liang ; Jim-Min Fang ; Jiun-Jie Shie ; Andrew H-J Wang | Structural basis of mercury- and zinc-conjugated complexes as SARS-CoV 3C-like protease inhibitors. |
| 001B63 (2008) |
Sara Cesarini [Italie] ; Andrea Spallarossa ; Angelo Ranise ; Paola Fossa ; Paolo La Colla ; Giuseppina Sanna ; Gabriella Collu ; Roberta Loddo | Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 1: Parallel synthesis, molecular modelling and structure-activity relationship studies on O-[2-(hetero)arylethyl]-N-phenylthiocarbamates. |
| 001B64 (2008) |
Sara Cesarini [Italie] ; Andrea Spallarossa ; Angelo Ranise ; Olga Bruno ; Paolo La Colla ; Barbara Secci ; Gabriella Collu ; Roberta Loddo | Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 2: Parallel synthesis, molecular modelling and structure-activity relationship studies on analogues of O-(2-phenylethyl)-N-phenylthiocarbamate. |
| 001B84 (2008) |
Jianmin Zhang [Canada] ; Carly Huitema ; Chunying Niu ; Jiang Yin ; Michael N G. James ; Lindsay D. Eltis ; John C. Vederas | Aryl methylene ketones and fluorinated methylene ketones as reversible inhibitors for severe acute respiratory syndrome (SARS) 3C-like proteinase. |
| 001B98 (2008) |
Yi-Ming Shao [Taïwan] ; Wen-Bin Yang [Taïwan] ; Tun-Hsun Kuo [Taïwan] ; Keng-Chang Tsai [Taïwan] ; Chun-Hung Lin [Taïwan] ; An-Suei Yang [Taïwan] ; Po-Huang Liang [Taïwan] ; Chi-Huey Wong [Taïwan, États-Unis] | Design, synthesis, and evaluation of trifluoromethyl ketones as inhibitors of SARS-CoV 3CL protease |
| 001C01 (2008) |
Prasenjit Mukherjee [États-Unis] ; Prashant Desai [États-Unis] ; Larry Ross [États-Unis] ; E. Lucile White [États-Unis] ; Mitchell A. Avery [États-Unis] | Structure-based virtual screening against SARS-3CLpro to identify novel non-peptidic hits |
| 001C06 (2008) |
Monica R. Loizzo [Italie] ; Antoine M. Saab ; Rosa Tundis ; Giancarlo A. Statti ; Francesco Menichini ; Ilaria Lampronti ; Roberto Gambari ; Jindrich Cinatl ; Hans Wilhelm Doerr | Phytochemical analysis and in vitro antiviral activities of the essential oils of seven Lebanon species. |
| 001C26 (2008) |
Carly Huitema [Canada] ; Jianmin Zhang ; Jiang Yin ; Michael N G. James ; John C. Vederas ; Lindsay D. Eltis | Heteroaromatic ester inhibitors of hepatitis A virus 3C proteinase: Evaluation of mode of action. |
| 001C30 (2008) |
Dale L. Barnard [États-Unis] ; Craig W. Day [États-Unis] ; Kevin Bailey [États-Unis] ; Matthew Heiner [États-Unis] ; Robert Montgomery [États-Unis] ; Larry Lauridsen [États-Unis] ; Kie-Hoon Jung [États-Unis] ; Joseph K.-K. Li [États-Unis] ; Paul K. S. Chan [République populaire de Chine] ; Robert W. Sidwell [États-Unis] | Is the anti-psychotic, 10-(3-(dimethylamino)propyl)phenothiazine (promazine), a potential drug with which to treat SARS infections? |
