Ident. | Authors (with country if any) | Title |
---|
000C12 (2004) |
Susan C. Baker [États-Unis] | Coronaviruses: from common colds to severe acute respiratory syndrome. |
000C30 (2004) |
Brian H. Harcourt [États-Unis] ; Dalia Jukneliene ; Amornrat Kanjanahaluethai ; John Bechill ; Kari M. Severson ; Catherine M. Smith ; Paul A. Rota ; Susan C. Baker | Identification of severe acute respiratory syndrome coronavirus replicase products and characterization of papain-like protease activity. |
001229 (2005) |
Arun K. Ghosh [États-Unis] ; Kai Xi ; Kiira Ratia ; Bernard D. Santarsiero ; Wentao Fu ; Brian H. Harcourt ; Paul A. Rota ; Susan C. Baker ; Michael E. Johnson ; Andrew D. Mesecar | Design and synthesis of peptidomimetic severe acute respiratory syndrome chymotrypsin-like protease inhibitors. |
001277 (2005) |
Naina Barretto ; Dalia Jukneliene ; Kiira Ratia ; Zhongbin Chen ; Andrew D. Mesecar ; Susan C. Baker | The Papain-Like Protease of Severe Acute Respiratory Syndrome Coronavirus Has Deubiquitinating Activity |
001439 (2006) |
Kiira Ratia [États-Unis] ; Kumar Singh Saikatendu ; Bernard D. Santarsiero ; Naina Barretto ; Susan C. Baker ; Raymond C. Stevens ; Andrew D. Mesecar | Severe acute respiratory syndrome coronavirus papain-like protease: structure of a viral deubiquitinating enzyme. |
001687 (2006) |
Naina Barretto [États-Unis] ; Dalia Jukneliene ; Kiira Ratia ; Zhongbin Chen ; Andrew D. Mesecar ; Susan C. Baker | Deubiquitinating activity of the SARS-CoV papain-like protease. |
001913 (2007) |
Zhongbin Chen ; Yanhua Wang ; Kiira Ratia ; Andrew D. Mesecar ; Keith D. Wilkinson ; Susan C. Baker | Proteolytic Processing and Deubiquitinating Activity of Papain-Like Proteases of Human Coronavirus NL63▿ |
001915 (2008) |
Valerie Grum-Tokars [États-Unis] ; Kiira Ratia ; Adrian Begaye ; Susan C. Baker ; Andrew D. Mesecar | Evaluating the 3C-like protease activity of SARS-Coronavirus: recommendations for standardized assays for drug discovery. |
001A50 (2007) |
Santhana G. Devaraj [États-Unis] ; Nan Wang ; Zhongbin Chen ; Zihong Chen ; Monica Tseng ; Naina Barretto ; Rongtuan Lin ; Clarence J. Peters ; Chien-Te K. Tseng ; Susan C. Baker ; Kui Li | Regulation of IRF-3-dependent innate immunity by the papain-like protease domain of the severe acute respiratory syndrome coronavirus. |
001A60 (2007) |
Arun K. Ghosh [États-Unis] ; Kai Xi [États-Unis] ; Valerie Grum-Tokars [États-Unis] ; Xiaoming Xu [États-Unis] ; Kiira Ratia [États-Unis] ; Wentao Fu [États-Unis] ; Katherine V. Houser [États-Unis] ; Susan C. Baker [États-Unis] ; Michael E. Johnson [États-Unis] ; Andrew D. Mesecar [États-Unis] | Structure-based design, synthesis, and biological evaluation of peptidomimetic SARS-CoV 3CLpro inhibitors |
001D48 (2008) |
Arun K. Ghosh [États-Unis] ; Gangli Gong [États-Unis] ; Valerie Grum-Tokars [États-Unis] ; Debbie C. Mulhearn [États-Unis] ; Susan C. Baker [États-Unis] ; Melissa Coughlin [États-Unis] ; Bellur S. Prabhakar [États-Unis] ; Katrina Sleeman [États-Unis] ; Michael E. Johnson [États-Unis] ; Andrew D. Mesecar [États-Unis] | Design, synthesis and antiviral efficacy of a series of potent chloropyridyl ester-derived SARS-CoV 3CLpro inhibitors |
001D66 (2008) |
Kiira Ratia [États-Unis] ; Scott Pegan ; Jun Takayama ; Katrina Sleeman ; Melissa Coughlin ; Surendranath Baliji ; Rima Chaudhuri ; Wentao Fu ; Bellur S. Prabhakar ; Michael E. Johnson ; Susan C. Baker ; Arun K. Ghosh ; Andrew D. Mesecar | A noncovalent class of papain-like protease/deubiquitinase inhibitors blocks SARS virus replication. |
001F75 (2009) |
Arun K. Ghosh [États-Unis] ; Jun Takayama [États-Unis] ; Yoann Aubin [États-Unis] ; Kiira Ratia [États-Unis] ; Rima Chaudhuri [États-Unis] ; Yahira Baez [États-Unis] ; Katrina Sleeman [États-Unis] ; Melissa Coughlin [États-Unis] ; Daniel B. Nichols [États-Unis] ; Debbie C. Mulhearn [États-Unis] ; Bellur S. Prabhakar [États-Unis] ; Susan C. Baker [États-Unis] ; Michael E. Johnson [États-Unis] ; Andrew D. Mesecar [États-Unis] | Structure-Based Design, Synthesis, and Biological Evaluation of a Series of Novel and Reversible Inhibitors for the Severe Acute Respiratory Syndrome-Coronavirus Papain-Like Protease |
001F76 (2006) |
Arun K. Ghosh [États-Unis] ; Kai Xi [États-Unis] ; Michael E. Johnson [États-Unis] ; Susan C. Baker [États-Unis] ; Andrew D. Mesecar [États-Unis] | Progress in Anti-SARS Coronavirus Chemistry, Biology and Chemotherapy |
002085 (2010) |
Mark A. Clementz [États-Unis] ; Zhongbin Chen ; Bridget S. Banach ; Yanhua Wang ; Li Sun ; Kiira Ratia ; Yahira M. Baez-Santos ; Jie Wang ; Jun Takayama ; Arun K. Ghosh ; Kui Li ; Andrew D. Mesecar ; Susan C. Baker | Deubiquitinating and interferon antagonism activities of coronavirus papain-like proteases. |
002151 (2010) |
Arun K. Ghosh [États-Unis] ; Jun Takayama [États-Unis] ; Kalapala Venkateswara Rao [États-Unis] ; Kiira Ratia [États-Unis] ; Rima Chaudhuri [États-Unis] ; Debbie C. Mulhearn [États-Unis] ; Hyun Lee [États-Unis] ; Daniel B. Nichols [États-Unis] ; Surendranath Baliji [États-Unis] ; Susan C. Baker [États-Unis] ; Michael E. Johnson [États-Unis] ; Andrew D. Mesecar [États-Unis] | Severe Acute Respiratory Syndrome-Coronavirus Papain-Like Novel Protease Inhibitors: Design, Synthesis, Protein-Ligand X-ray Structure and Biological Evaluation |
002454 (2012) |
Li Sun [République populaire de Chine] ; Yaling Xing ; Xiaojuan Chen ; Yang Zheng ; Yudong Yang ; Daniel B. Nichols ; Mark A. Clementz ; Bridget S. Banach ; Kui Li ; Susan C. Baker ; Zhongbin Chen | Coronavirus papain-like proteases negatively regulate antiviral innate immune response through disruption of STING-mediated signaling. |
002590 (2012) |
Hatem A. Elshabrawy [États-Unis] ; Melissa M. Coughlin ; Susan C. Baker ; Bellur S. Prabhakar | Human monoclonal antibodies against highly conserved HR1 and HR2 domains of the SARS-CoV spike protein are more broadly neutralizing. |
002596 (2013) |
Jon Jacobs [États-Unis] ; Valerie Grum-Tokars ; Ya Zhou ; Mark Turlington ; S Adrian Saldanha ; Peter Chase ; Aimee Eggler ; Eric S. Dawson ; Yahira M. Baez-Santos ; Sakshi Tomar ; Anna M. Mielech ; Susan C. Baker ; Craig W. Lindsley ; Peter Hodder ; Andrew Mesecar ; Shaun R. Stauffer | Discovery, synthesis, and structure-based optimization of a series of N-(tert-butyl)-2-(N-arylamido)-2-(pyridin-3-yl) acetamides (ML188) as potent noncovalent small molecule inhibitors of the severe acute respiratory syndrome coronavirus (SARS-CoV) 3CL protease. |
002741 (2013) |
Andy Kilianski [États-Unis] ; Anna M. Mielech ; Xufang Deng ; Susan C. Baker | Assessing activity and inhibition of Middle East respiratory syndrome coronavirus papain-like and 3C-like proteases using luciferase-based biosensors. |
002786 (2014) |
Andy Kilianski [États-Unis] ; Susan C. Baker [États-Unis] | Cell-based antiviral screening against coronaviruses: developing virus-specific and broad-spectrum inhibitors. |