Ident. | Authors (with country if any) | Title |
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001007 (2016) |
Vathan Kumar [Taïwan] ; Kian-Pin Tan [Taïwan] ; Ying-Ming Wang [Taïwan] ; Sheng-Wei Lin [Taïwan] ; Po-Huang Liang [Taïwan] | Identification, synthesis and evaluation of SARS-CoV and MERS-CoV 3C-like protease inhibitors. |
001050 (2016) |
Bao-Long Chen [République populaire de Chine] ; Ya-Jing Wang [République populaire de Chine] ; Hong Guo [République populaire de Chine] ; Guang-Yao Zeng [République populaire de Chine] | Design, synthesis, and biological evaluation of crenatoside analogues as novel influenza neuraminidase inhibitors. |
001051 (2016) |
Qing Meng [République populaire de Chine] ; Xuwang Chen [République populaire de Chine] ; Dongwei Kang [République populaire de Chine] ; Boshi Huang [République populaire de Chine] ; Wenxin Li [République populaire de Chine] ; Peng Zhan [République populaire de Chine] ; Dirk Daelemans [Belgique] ; Erik De Clercq [Belgique] ; Christophe Pannecouque [Belgique] ; Xinyong Liu [République populaire de Chine] | Design, synthesis and evaluation of novel HIV-1 NNRTIs with dual structural conformations targeting the entrance channel of the NNRTI binding pocket. |
001052 (2016) |
Jiapei Yang [République populaire de Chine] ; Wenmin Chen [République populaire de Chine] ; Dongwei Kang [République populaire de Chine] ; Xueyi Lu [République populaire de Chine] ; Xiao Li [République populaire de Chine] ; Zhaoqiang Liu [République populaire de Chine] ; Boshi Huang [République populaire de Chine] ; Dirk Daelemans [Belgique] ; Christophe Pannecouque [Belgique] ; Erik De Clercq [Belgique] ; Peng Zhan [République populaire de Chine] ; Xinyong Liu [République populaire de Chine] | Design, synthesis and anti-HIV evaluation of novel diarylpyridine derivatives targeting the entrance channel of NNRTI binding pocket. |
001231 (2015) |
Yuanyuan Cao [République populaire de Chine] ; Yu Zhang [République populaire de Chine] ; Shaotong Wu [République populaire de Chine] ; Quanzhi Yang [République populaire de Chine] ; Xuefeng Sun [République populaire de Chine] ; Jianxiong Zhao [République populaire de Chine] ; Fen Pei [République populaire de Chine] ; Ying Guo [République populaire de Chine] ; Chao Tian [République populaire de Chine] ; Zhili Zhang [République populaire de Chine] ; Haining Wang [République populaire de Chine] ; Liying Ma [République populaire de Chine] ; Junyi Liu [République populaire de Chine] ; Xiaowei Wang [République populaire de Chine] | Synthesis and biological evaluation of pyridinone analogues as novel potent HIV-1 NNRTIs. |
001233 (2015) |
Zan Li [République populaire de Chine] ; Zhaoliang Li [République populaire de Chine] ; Yunwei Lin [République populaire de Chine] ; Zhaoqing Meng [République populaire de Chine] ; Gang Ding [République populaire de Chine] ; Liang Cao [République populaire de Chine] ; Na Li [République populaire de Chine] ; Wenjun Liu [République populaire de Chine] ; Wei Xiao [République populaire de Chine] ; Xiaoming Wu [République populaire de Chine] ; Jinyi Xu [République populaire de Chine] | Synthesis and Biological Evaluation of Strictosamide Derivatives with Improved Antiviral and Antiproliferative Activities. |
001234 (2015) |
Nobuko Mibu ; Kazumi Yokomizo ; Hatsumi Aki ; Norimasa Ota ; Hiroyuki Fujii ; Ai Yuzuriha ; Shiori Saneyoshi ; Aoi Tanaka ; Airi Koga ; Jianrong Zhou ; Takeshi Miyata ; Kunihiro Sumoto | Synthesis and Antiviral Evaluation of Some C(3)-Symmetrical Trialkoxy-Substituted 1,3,5-Triazines and Their Molecular Geometry. |
001291 (2015) |
Yong Zhao [République populaire de Chine] ; Chang-An Geng [République populaire de Chine] ; Hao Chen [République populaire de Chine] ; Yun-Bao Ma [République populaire de Chine] ; Xiao-Yan Huang [République populaire de Chine] ; Tuan-Wu Cao [République populaire de Chine] ; Kang He [République populaire de Chine] ; Hao Wang [République populaire de Chine] ; Xue-Mei Zhang [République populaire de Chine] ; Ji-Jun Chen [République populaire de Chine] | Isolation, synthesis and anti-hepatitis B virus evaluation of p-hydroxyacetophenone derivatives from Artemisia capillaris. |
001319 (2015) |
Linda A. Selvey ; Catarina Antão ; Robert Hall | Evaluation of Border Entry Screening for Infectious Diseases in Humans |
001335 (2015) |
Sheng Liu [République populaire de Chine] ; Wanxing Wei [République populaire de Chine] ; Yubin Li [République populaire de Chine] ; Xu Liu [République populaire de Chine] ; Xiaoji Cao [République populaire de Chine] ; Kechan Lei [République populaire de Chine] ; Min Zhou [République populaire de Chine] | Design, synthesis, biological evaluation and molecular docking studies of phenylpropanoid derivatives as potent anti-hepatitis B virus agents. |
001336 (2015) |
Hannah L. Peters [États-Unis] ; Dirk Jochmans [Belgique] ; Adriaan H. De Wilde [Pays-Bas] ; Clara C. Posthuma [Pays-Bas] ; Eric J. Snijder [Pays-Bas] ; Johan Neyts [Belgique] ; Katherine L. Seley-Radtke [États-Unis] | Design, synthesis and evaluation of a series of acyclic fleximer nucleoside analogues with anti-coronavirus activity. |
001337 (2015) |
Li-Jun Wang ; Hao Chen ; Yun-Bao Ma ; Xiao-Yan Huang ; Chang-An Geng ; Xue-Mei Zhang ; Ji-Jun Chen [République populaire de Chine] | Design, synthesis and biological evaluation of caudatin analogs as potent hepatitis B virus inhibitors. |
001338 (2015) |
Tao Liu [République populaire de Chine] ; Boshi Huang [République populaire de Chine] ; Ye Tian [République populaire de Chine] ; Xin Liang [République populaire de Chine] ; Hong Liu [République populaire de Chine] ; Huiqing Liu [République populaire de Chine] ; Peng Zhan [République populaire de Chine] ; Erik De Clercq [Belgique] ; Christophe Pannecouque [Belgique] ; Xinyong Liu [République populaire de Chine] | Design, Synthesis, and Biological Evaluation of Novel 4-Aminopiperidinyl-linked 3,5-Disubstituted-1,2,6-thiadiazine-1,1-dione Derivatives as HIV-1 NNRTIs. |
001412 (2015) |
Jingjing Gao [République populaire de Chine] ; Xianjin Luo [République populaire de Chine] ; Yuhuan Li [République populaire de Chine] ; Rongmei Gao [République populaire de Chine] ; Haifeng Chen [République populaire de Chine] ; Dingjue Ji [République populaire de Chine] | Synthesis and Biological Evaluation of 2‐oxo‐pyrazine‐3‐carboxamide‐yl Nucleoside Analogues and Their Epimers as Inhibitors of Influenza A Viruses |
001518 (2014) |
Nicolas Primas [France] ; Peggy Suzanne [France] ; Pierre Verhaeghe [France] ; Sébastien Hutter [France] ; Charline Kieffer [France] ; Michèle Laget [France] ; Anita Cohen [France] ; Julie Broggi [France] ; Jean-Charles Lancelot [France] ; Aurélien Lesnard [France] ; Patrick Dallemagne [France] ; Pascal Rathelot [France] ; Sylvain Rault [France] ; Patrice Vanelle [France] ; Nadine Azas [France] | Synthesis and in vitro evaluation of 4-trichloromethylpyrrolo[1,2-a]quinoxalines as new antiplasmodial agents |
001530 (2014) |
Yahira M. Báez-Santos [États-Unis] ; Scott J. Barraza ; Michael W. Wilson ; Michael P. Agius ; Anna M. Mielech ; Nicole M. Davis ; Susan C. Baker ; Scott D. Larsen ; Andrew D. Mesecar | X-ray structural and biological evaluation of a series of potent and highly selective inhibitors of human coronavirus papain-like proteases. |
001557 (2014) |
Hao Chen [République populaire de Chine] ; Yun-Bao Ma [République populaire de Chine] ; Xiao-Yan Huang [République populaire de Chine] ; Chang-An Geng [République populaire de Chine] ; Yong Zhao [République populaire de Chine] ; Li-Jun Wang [République populaire de Chine] ; Rui-Hua Guo [République populaire de Chine] ; Wen-Juan Liang [République populaire de Chine] ; Xue-Mei Zhang [République populaire de Chine] ; Ji-Jun Chen [République populaire de Chine] | Synthesis, structure-activity relationships and biological evaluation of dehydroandrographolide and andrographolide derivatives as novel anti-hepatitis B virus agents. |
001558 (2014) |
Reham A I. Abou-Elkhair [Égypte] ; Ahmed H. Moustafa [Égypte] ; Abdelfattah Z. Haikal [Égypte] ; Ahmed M. Ibraheem [Égypte] | Synthesis and biological evaluation of 2-oxonicotinonitriles and 2-oxonicotinonitrile based nucleoside analogues. |
001652 (2014) |
Adeyemi O. Adedeji [États-Unis] ; Kamalendra Singh [États-Unis] ; Ademola Kassim [États-Unis] ; Christopher M. Coleman [États-Unis] ; Ruth Elliott [États-Unis] ; Susan R. Weiss [États-Unis] ; Matthew B. Frieman [États-Unis] ; Stefan G. Sarafianos [États-Unis] | Evaluation of SSYA10-001 as a replication inhibitor of severe acute respiratory syndrome, mouse hepatitis, and Middle East respiratory syndrome coronaviruses. |
001667 (2014) |
Zhaoqiang Liu [République populaire de Chine] ; Wenmin Chen [République populaire de Chine] ; Peng Zhan [République populaire de Chine] ; Erik De Clercq [Belgique] ; Christophe Pannecouque [Belgique] ; Xinyong Liu [République populaire de Chine] | Design, synthesis and anti-HIV evaluation of novel diarylnicotinamide derivatives (DANAs) targeting the entrance channel of the NNRTI binding pocket through structure-guided molecular hybridization. |
001700 (2014) |
Xiao Li [République populaire de Chine] ; Xueyi Lu [République populaire de Chine] ; Wenmin Chen [République populaire de Chine] ; Huiqing Liu [République populaire de Chine] ; Peng Zhan [République populaire de Chine] ; Christophe Pannecouque [Belgique] ; Jan Balzarini [Belgique] ; Erik De Clercq [Belgique] ; Xinyong Liu [République populaire de Chine] | Arylazolyl(azinyl)thioacetanilides. Part 16: Structure-based bioisosterism design, synthesis and biological evaluation of novel pyrimidinylthioacetanilides as potent HIV-1 inhibitors. |