Ident. | Authors (with country if any) | Title |
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000C31 (2018) |
Cy V. Credille [États-Unis] ; Benjamin L. Dick [États-Unis] ; Christine N. Morrison [États-Unis] ; Ryjul W. Stokes [États-Unis] ; Rebecca N. Adamek [États-Unis] ; Nicholas C. Wu [États-Unis] ; Ian A. Wilson [États-Unis] ; Seth M. Cohen [États-Unis] | Structure-Activity Relationships in Metal-Binding Pharmacophores for Influenza Endonuclease. |
000C90 (2018) |
Min-Han Lin [Taïwan] ; David C. Moses [Taïwan] ; Chih-Hua Hsieh [Taïwan] ; Shu-Chun Cheng [Taïwan] ; Yau-Hung Chen [Taïwan] ; Chiao-Yin Sun [Taïwan] ; Chi-Yuan Chou [Taïwan] | Disulfiram can inhibit MERS and SARS coronavirus papain-like proteases via different modes. |
000D48 (2017) |
Wahiba Aouadi [France] ; Cécilia Eydoux [France] ; Bruno Coutard [France] ; Baptiste Martin [France] ; Françoise Debart [France] ; Jean Jacques Vasseur [France] ; Jean Marie Contreras [France] ; Christophe Morice [France] ; Gilles Quérat [France] ; Marie-Louise Jung [France] ; Bruno Canard [France] ; Jean-Claude Guillemot [France] ; Etienne Decroly [France] | Toward the identification of viral cap-methyltransferase inhibitors by fluorescence screening assay |
000E83 (2017) |
Jin-Moo Lee [Corée du Sud] ; Jin-Beom Cho [Corée du Sud] ; Hee-Chul Ahn [Corée du Sud] ; Woong Jung [Corée du Sud] ; Yong-Joo Jeong [Corée du Sud] | A Novel Chemical Compound for Inhibition of SARS Coronavirus Helicase. |
001007 (2016) |
Vathan Kumar [Taïwan] ; Kian-Pin Tan [Taïwan] ; Ying-Ming Wang [Taïwan] ; Sheng-Wei Lin [Taïwan] ; Po-Huang Liang [Taïwan] | Identification, synthesis and evaluation of SARS-CoV and MERS-CoV 3C-like protease inhibitors. |
001049 (2016) |
Sheng Liu [République populaire de Chine] ; Yubin Li [République populaire de Chine] ; Wanxing Wei [République populaire de Chine] ; Kuiwu Wang [République populaire de Chine] ; Lisheng Wang [République populaire de Chine] ; Jianyi Wang [République populaire de Chine] | Design, synthesis, molecular docking studies and anti-HBV activity of phenylpropanoid derivatives. |
001089 (2016) |
Hanjun Zhao [République populaire de Chine] ; Jie Zhou [République populaire de Chine] ; Ke Zhang [République populaire de Chine] ; Hin Chu [République populaire de Chine] ; Dabin Liu [République populaire de Chine] ; Vincent Kwok-Man Poon [République populaire de Chine] ; Chris Chung-Sing Chan [République populaire de Chine] ; Ho-Chuen Leung [République populaire de Chine] ; Ng Fai [République populaire de Chine] ; Yong-Ping Lin [République populaire de Chine] ; Anna Jin-Xia Zhang [République populaire de Chine] ; Dong-Yan Jin [République populaire de Chine] ; Kwok-Yung Yuen [République populaire de Chine] ; Bo-Jian Zheng [République populaire de Chine] | A novel peptide with potent and broad-spectrum antiviral activities against multiple respiratory viruses |
001304 (2015) |
Jin-Beom Cho [Corée du Sud] ; Jin-Moo Lee [Corée du Sud] ; Hee-Chul Ahn [Corée du Sud] ; Yong-Joo Jeong [Corée du Sud] | Identification of a Novel Small Molecule Inhibitor Against SARS Coronavirus Helicase. |
001529 (2014) |
Ying Sun [République populaire de Chine] ; Zidao Wang [République populaire de Chine] ; Jiali Tao [République populaire de Chine] ; Yi Wang [République populaire de Chine] ; Andong Wu [République populaire de Chine] ; Ziwen Yang [République populaire de Chine] ; Kaimei Wang [République populaire de Chine] ; Liqiao Shi [République populaire de Chine] ; Yu Chen [République populaire de Chine] ; Deyin Guo [République populaire de Chine] | Yeast-based assays for the high-throughput screening of inhibitors of coronavirus RNA cap guanine-N7-methyltransferase. |
001563 (2014) |
K B Wong [Hong Kong] ; D C C. Wan [Hong Kong] ; H F Chow [Hong Kong] | Substrate specificity and rational design of peptidomimetic inhibitors for SARS coronavirus main protease. |
001594 (2014) |
C P Chuck [Hong Kong] ; Z H Ke [Hong Kong] ; C. Chen [Hong Kong] ; D C C. Wan [Hong Kong] ; H F Chow [Hong Kong] ; K B Wong [Hong Kong] | Profiling of substrate-specificity and rational design of broad-spectrum peptidomimetic inhibitors for main proteases of coronaviruses. |
001604 (2014) |
Yeong Hun Song ; Dae Wook Kim ; Marcus John Curtis-Long ; Heung Joo Yuk ; Yan Wang ; Ningning Zhuang ; Kon Ho Lee ; Kwon Seok Jeon ; Ki Hun Park | Papain-like protease (PLpro) inhibitory effects of cinnamic amides from Tribulus terrestris fruits. |
001652 (2014) |
Adeyemi O. Adedeji [États-Unis] ; Kamalendra Singh [États-Unis] ; Ademola Kassim [États-Unis] ; Christopher M. Coleman [États-Unis] ; Ruth Elliott [États-Unis] ; Susan R. Weiss [États-Unis] ; Matthew B. Frieman [États-Unis] ; Stefan G. Sarafianos [États-Unis] | Evaluation of SSYA10-001 as a replication inhibitor of severe acute respiratory syndrome, mouse hepatitis, and Middle East respiratory syndrome coronaviruses. |
001961 (2013) |
Pillaiyar Thanigaimalai [Japon] ; Sho Konno ; Takehito Yamamoto ; Yuji Koiwai ; Akihiro Taguchi ; Kentaro Takayama ; Fumika Yakushiji ; Kenichi Akaji ; Shen-En Chen ; Aurash Naser-Tavakolian ; Arne Schön ; Ernesto Freire ; Yoshio Hayashi | Development of potent dipeptide-type SARS-CoV 3CL protease inhibitors with novel P3 scaffolds: design, synthesis, biological evaluation, and docking studies. |
001966 (2013) |
Tao Liu [République populaire de Chine] ; Zhiyong Weng [République populaire de Chine] ; Xiaowu Dong [République populaire de Chine] ; Linjie Chen [République populaire de Chine] ; Ling Ma [République populaire de Chine] ; Shan Cen [République populaire de Chine] ; Naiming Zhou [République populaire de Chine] ; Yongzhou Hu [République populaire de Chine] | Design, Synthesis and Biological Evaluation of Novel Piperazine Derivatives as CCR5 Antagonists |
001C54 (2012) |
Adeyemi O. Adedeji [États-Unis] ; Kamalendra Singh ; Nicholas E. Calcaterra ; Marta L. Dediego ; Luis Enjuanes ; Susan Weiss ; Stefan G. Sarafianos | Severe acute respiratory syndrome coronavirus replication inhibitor that interferes with the nucleic acid unwinding of the viral helicase. |
001D21 (2012) |
Thi Thanh Hanh Nguyen [Corée du Sud] ; Hye-Jin Woo ; Hee-Kyoung Kang ; Van Dao Nguyen ; Young-Min Kim ; Do-Won Kim ; Sul-Ah Ahn ; Yongmei Xia ; Doman Kim | Flavonoid-mediated inhibition of SARS coronavirus 3C-like protease expressed in Pichia pastoris. |
002010 (2011) |
Qiaoli Li [République populaire de Chine] ; Zhenhuan Zhao ; Dihan Zhou ; Yaoqing Chen ; Wei Hong ; Luyang Cao ; Jingyi Yang ; Yan Zhang ; Wei Shi ; Zhijian Cao ; Yingliang Wu ; Huimin Yan ; Wenxin Li | Virucidal activity of a scorpion venom peptide variant mucroporin-M1 against measles, SARS-CoV and influenza H5N1 viruses. |
002011 (2011) |
Thi Thanh Hanh Nguyen [Corée du Sud] ; Hwa-Ja Ryu ; Se-Hoon Lee ; Soonwook Hwang ; Vincent Breton ; Joon Haeng Rhee ; Doman Kim | Virtual screening identification of novel severe acute respiratory syndrome 3C-like protease inhibitors and in vitro confirmation. |
002093 (2011) |
Prasenjit Mukherjee ; Falgun Shah ; Prashant Desai ; Mitchell Avery | Inhibitors of SARS-3CLpro: Virtual Screening, Biological Evaluation and Molecular Dynamics Simulation Studies |
002109 (2011) |
Xiaoqing Chen [République populaire de Chine] ; Zhongxia Wang ; Ziying Yang ; Jingjing Wang ; Yunxia Xu ; Ren-Xiang Tan ; Erguang Li | Houttuynia cordata blocks HSV infection through inhibition of NF-κB activation. |