Ident. | Authors (with country if any) | Title |
---|
000C90 (2018) |
Min-Han Lin [Taïwan] ; David C. Moses [Taïwan] ; Chih-Hua Hsieh [Taïwan] ; Shu-Chun Cheng [Taïwan] ; Yau-Hung Chen [Taïwan] ; Chiao-Yin Sun [Taïwan] ; Chi-Yuan Chou [Taïwan] | Disulfiram can inhibit MERS and SARS coronavirus papain-like proteases via different modes. |
000F42 (2016) |
Bo Su [République populaire de Chine] ; Chunlong Cai [République populaire de Chine] ; Meng Deng [République populaire de Chine] ; Qingmin Wang [République populaire de Chine] | Spatial Configuration and Three-Dimensional Conformation Directed Design, Synthesis, Antiviral Activity, and Structure-Activity Relationships of Phenanthroindolizidine Analogues. |
001272 (2015) |
Jun-Li Yang [Corée du Sud] ; Thi-Kim-Quy Ha ; Basanta Dhodary ; Euisun Pyo ; Ngoc Hieu Nguyen ; Hyomoon Cho ; Eunhee Kim ; Won Keun Oh | Oleanane triterpenes from the flowers of Camellia japonica inhibit porcine epidemic diarrhea virus (PEDV) replication. |
001530 (2014) |
Yahira M. Báez-Santos [États-Unis] ; Scott J. Barraza ; Michael W. Wilson ; Michael P. Agius ; Anna M. Mielech ; Nicole M. Davis ; Susan C. Baker ; Scott D. Larsen ; Andrew D. Mesecar | X-ray structural and biological evaluation of a series of potent and highly selective inhibitors of human coronavirus papain-like proteases. |
001705 (2014) |
Dustin B. Ritchie [Canada] ; Jingchyuan Soong ; William K A. Sikkema ; Michael T. Woodside | Anti-frameshifting ligand reduces the conformational plasticity of the SARS virus pseudoknot. |
001904 (2013) |
Sivakoteswara Rao Mandadapu [États-Unis] ; Pathum M. Weerawarna ; Allan M. Prior ; Roxanne Adeline Z. Uy ; Sridhar Aravapalli ; Kevin R. Alliston ; Gerald H. Lushington ; Yunjeong Kim ; Duy H. Hua ; Kyeong-Ok Chang ; William C. Groutas | Macrocyclic inhibitors of 3C and 3C-like proteases of picornavirus, norovirus, and coronavirus. |
001964 (2013) |
Pillaiyar Thanigaimalai [Japon] ; Sho Konno [Japon] ; Takehito Yamamoto [Japon] ; Yuji Koiwai [Japon] ; Akihiro Taguchi [Japon] ; Kentaro Takayama [Japon] ; Fumika Yakushiji [Japon] ; Kenichi Akaji [Japon] ; Yoshiaki Kiso [Japon] ; Yuko Kawasaki [États-Unis] ; Shen-En Chen [États-Unis] ; Aurash Naser-Tavakolian [États-Unis] ; Arne Schön [États-Unis] ; Ernesto Freire [États-Unis] ; Yoshio Hayashi [Japon] | Design, synthesis, and biological evaluation of novel dipeptide-type SARS-CoV 3CL protease inhibitors: Structure–activity relationship study |
002436 (2010) |
Iou-Jiun Kang [République populaire de Chine] ; Li-Wen Wang ; Teng-Kuang Yeh ; Chung-Chi Lee ; Yen-Chun Lee ; Sheng-Ju Hsu ; Yen-Shian Wu ; Jing-Chyi Wang ; Yu-Sheng Chao ; Andrew Yueh ; Jyh-Haur Chern | Synthesis, activity, and pharmacokinetic properties of a series of conformationally-restricted thiourea analogs as novel hepatitis C virus inhibitors. |
002A84 (2009) |
Fumiaki N. Ishikawa [États-Unis] ; Hsiao-Kang Chang ; Marco Curreli ; Hsiang-I Liao ; C Anders Olson ; Po-Chiang Chen ; Rui Zhang ; Richard W. Roberts ; Ren Sun ; Richard J. Cote ; Mark E. Thompson ; Chongwu Zhou | Label-free, electrical detection of the SARS virus N-protein with nanowire biosensors utilizing antibody mimics as capture probes. |
003511 (2008) |
Arun K. Ghosh [États-Unis] ; GANGLI GONG [États-Unis] ; Valerie Grum-Tokars [États-Unis] ; Debbie C. Mulhearn [États-Unis] ; Susan C. Baker [États-Unis] ; Melissa Coughlin [États-Unis] ; Bellur S. Prabhakar [États-Unis] ; Katrina Sleeman [États-Unis] ; Michael E. Johnson [États-Unis] ; Andrew D. Mesecar [États-Unis] | Design, synthesis and antiviral efficacy of a series of potent chloropyridyl ester-derived SARS-CoV 3CLpro inhibitors |
003552 (2007) |
S-Q Wang [République populaire de Chine] ; Q-S Du ; K. Zhao ; A-X Li ; D-Q Wei ; K-C Chou | Virtual screening for finding natural inhibitor against cathepsin-L for SARS therapy. |
003586 (2007) |
Yi-Ming Shao [République populaire de Chine] ; Wen-Bin Yang ; Hung-Pin Peng ; Min-Feng Hsu ; Keng-Chang Tsai ; Tun-Hsun Kuo ; Andrew H-J Wang ; Po-Huang Liang ; Chun-Hung Lin ; An-Suei Yang ; Chi-Huey Wong | Structure-based design and synthesis of highly potent SARS-CoV 3CL protease inhibitors. |
003672 (2007) |
Qi-Shi Du [République populaire de Chine] ; Hao Sun ; Kuo-Chen Chou | Inhibitor design for SARS coronavirus main protease based on "distorted key theory". |
003743 (2007) |
Daniel R. Beniac [Canada] ; Shauna L. Devarennes ; Anton Andonov ; Runtao He ; Tim F. Booth | Conformational reorganization of the SARS coronavirus spike following receptor binding: implications for membrane fusion. |
003B21 (2007) |
Masahiro Ikejiri [Japon] ; Masayuki Saijo [Japon] ; Shigeru Morikawa [Japon] ; Shuetsu Fukushi [Japon] ; Tetsuya Mizutani [Japon] ; Ichiro Kurane [Japon] ; Tokumi Maruyama [Japon] | Synthesis and biological evaluation of nucleoside analogues having 6-chloropurine as anti-SARS-CoV agents |
003B49 (2007) |
Pedro Serrano [États-Unis] ; Margaret A. Johnson [États-Unis] ; Marcius S. Almeida [États-Unis] ; Reto Horst [États-Unis] ; Torsten Herrmann [Suisse] ; Jeremiah S. Joseph [États-Unis] ; Benjamin W. Neuman [États-Unis] ; Vanitha Subramanian [États-Unis] ; Kumar S. Saikatendu [États-Unis] ; Michael J. Buchmeier [États-Unis] ; Raymond C. Stevens [États-Unis] ; Peter Kuhn [États-Unis] ; Kurt Wüthrich [États-Unis] | Nuclear magnetic resonance structure of the N-terminal domain of nonstructural protein 3 from the severe acute respiratory syndrome coronavirus |
003B80 (2007) |
Jeremiah S. Joseph [États-Unis] ; KUMAR SINGH SAIKATENDU [États-Unis] ; Vanitha Subramanian [États-Unis] ; Benjamin W. Neuman [États-Unis] ; Michael J. Buchmeier [États-Unis] ; Raymond C. Stevens [États-Unis] ; Peter Kuhn [États-Unis] | Crystal structure of a monomeric form of severe acute respiratory syndrome coronavirus endonuclease nspl5 suggests a role for hexamerization as an allosteric switch |
003B93 (2007) |
Masahiro Ikejiri [Japon] ; Takayuki Ohshima [Japon] ; Keizo Kato [Japon] ; Masaaki Toyama [Japon] ; Takayuki Murata [Japon] ; Kunitada Shimotohno [Japon] ; Tokumi Maruyama [Japon] | 5'-O-Masked 2'-deoxyadenosine analogues as lead compounds for hepatitis C virus (HCV) therapeutic agents |
003C91 (2006) |
Rolf Hilgenfeld [Allemagne] ; Kanchan Anand ; Jeroen R. Mesters ; Zihe Rao ; Xu Shen ; Hualiang Jiang ; Jinzhi Tan ; Koen H G. Verschueren | Structure and dynamics of SARS coronavirus main proteinase (Mpro). |
003F20 (2006) |
Eric Assen B. Kantchev [République populaire de Chine] ; Chung-Chieh Chang ; Ding-Kwo Chang | Direct Fmoc/tert-Bu solid phase synthesis of octamannosyl polylysine dendrimer-peptide conjugates. |
004862 (2005) |
Zakaria A. Almsherqi [Singapour] ; Craig S. Mclachlan ; Peter Mossop ; Kèvin Knoops ; Yuru Deng | Direct template matching reveals a host subcellular membrane gyroid cubic structure that is associated with SARS virus. |