| Ident. | Authors (with country if any) | Title |
|---|
| 000B45 (2019) |
Kouji Ohnishi [Japon] ; Yasunao Hattori [Japon] ; Kazuya Kobayashi [Japon] ; Kenichi Akaji [Japon] | Evaluation of a non-prime site substituent and warheads combined with a decahydroisoquinolin scaffold as a SARS 3CL protease inhibitor. |
| 001071 (2016) |
Ji-Young Park [Corée du Sud] ; Jin-A Ko [Corée du Sud] ; Dae Wook Kim ; Young Min Kim [Corée du Sud] ; Hyung-Jun Kwon [Corée du Sud] ; Hyung Jae Jeong [Corée du Sud] ; Cha Young Kim [Corée du Sud] ; Ki Hun Park ; Woo Song Lee [Corée du Sud] ; Young Bae Ryu [Corée du Sud] | Chalcones isolated from Angelica keiskei inhibit cysteine proteases of SARS-CoV. |
| 001213 (2015) |
Kai-Wen Cheng [Taïwan] ; Shu-Chun Cheng [Taïwan] ; Wei-Yi Chen [Taïwan] ; Min-Han Lin [Taïwan] ; Shang-Ju Chuang [Taïwan] ; I-Hsin Cheng [Taïwan] ; Chiao-Yin Sun [Taïwan] ; Chi-Yuan Chou [Taïwan] | Thiopurine analogs and mycophenolic acid synergistically inhibit the papain-like protease of Middle East respiratory syndrome coronavirus. |
| 001269 (2015) |
Michael Berry [Afrique du Sud] ; Burtram C. Fielding [Afrique du Sud] ; Junaid Gamieldien [Afrique du Sud] | Potential Broad Spectrum Inhibitors of the Coronavirus 3CLpro: A Virtual Screening and Structure-Based Drug Design Study. |
| 001530 (2014) |
Yahira M. Báez-Santos [États-Unis] ; Scott J. Barraza ; Michael W. Wilson ; Michael P. Agius ; Anna M. Mielech ; Nicole M. Davis ; Susan C. Baker ; Scott D. Larsen ; Andrew D. Mesecar | X-ray structural and biological evaluation of a series of potent and highly selective inhibitors of human coronavirus papain-like proteases. |
| 001543 (2014) |
Yahira M. Báez-Santos ; Sarah E. St. John ; Andrew D. Mesecar | The SARS-coronavirus papain-like protease: Structure, function and inhibition by designed antiviral compounds |
| 001604 (2014) |
Yeong Hun Song ; Dae Wook Kim ; Marcus John Curtis-Long ; Heung Joo Yuk ; Yan Wang ; Ningning Zhuang ; Kon Ho Lee ; Kwon Seok Jeon ; Ki Hun Park | Papain-like protease (PLpro) inhibitory effects of cinnamic amides from Tribulus terrestris fruits. |
| 001960 (2013) |
Ji-Young Park [Corée du Sud] ; Jang Hoon Kim ; Jung Min Kwon ; Hyung-Jun Kwon ; Hyung Jae Jeong ; Young Min Kim ; Doman Kim ; Woo Song Lee ; Young Bae Ryu | Dieckol, a SARS-CoV 3CL(pro) inhibitor, isolated from the edible brown algae Ecklonia cava. |
| 001964 (2013) |
Pillaiyar Thanigaimalai [Japon] ; Sho Konno [Japon] ; Takehito Yamamoto [Japon] ; Yuji Koiwai [Japon] ; Akihiro Taguchi [Japon] ; Kentaro Takayama [Japon] ; Fumika Yakushiji [Japon] ; Kenichi Akaji [Japon] ; Yoshiaki Kiso [Japon] ; Yuko Kawasaki [États-Unis] ; Shen-En Chen [États-Unis] ; Aurash Naser-Tavakolian [États-Unis] ; Arne Schön [États-Unis] ; Ernesto Freire [États-Unis] ; Yoshio Hayashi [Japon] | Design, synthesis, and biological evaluation of novel dipeptide-type SARS-CoV 3CL protease inhibitors: Structure–activity relationship study |
| 001C44 (2012) |
Ji-Young Park [Corée du Sud] ; Jang Hoon Kim ; Young Min Kim ; Hyung Jae Jeong ; Dae Wook Kim ; Ki Hun Park ; Hyung-Jun Kwon ; Su-Jin Park ; Woo Song Lee ; Young Bae Ryu | Tanshinones as selective and slow-binding inhibitors for SARS-CoV cysteine proteases. |
| 001F62 (2012) |
Miyuki Kawase [Japon] ; Kazuya Shirato [Japon] ; Lia Van Der Hoek [Pays-Bas] ; Fumihiro Taguchi [Japon] ; Shutoku Matsuyama [Japon] | Simultaneous Treatment of Human Bronchial Epithelial Cells with Serine and Cysteine Protease Inhibitors Prevents Severe Acute Respiratory Syndrome Coronavirus Entry |
| 001F64 (2012) |
Martha Schneider [Allemagne] ; Kerstin Ackermann [Allemagne] ; Melissa Stuart [États-Unis] ; Claudia Wex [Allemagne] ; Ulrike Protzer [Allemagne] ; Hermann M. Sch Tzl [Allemagne, États-Unis] ; Sabine Gilch [Allemagne, États-Unis] | Severe Acute Respiratory Syndrome Coronavirus Replication Is Severely Impaired by MG132 due to Proteasome-Independent Inhibition of M-Calpain |
| 002566 (2010) |
Falgun Shah [États-Unis] ; Prasenjit Mukherjee ; Prashant Desai ; Mitchell Avery | Computational approaches for the discovery of cysteine protease inhibitors against malaria and SARS. |
| 002587 (2010) |
Parag P. Shah [États-Unis] ; Tianhua Wang ; Rachel L. Kaletsky ; Michael C. Myers ; Jeremy E. Purvis ; Huiyan Jing ; Donna M. Huryn ; Doron C. Greenbaum ; Amos B. Smith ; Paul Bates ; Scott L. Diamond | A small-molecule oxocarbazate inhibitor of human cathepsin L blocks severe acute respiratory syndrome and ebola pseudotype virus infection into human embryonic kidney 293T cells. |
| 002A10 (2009) |
Cheng-Chung Lee [Taïwan] ; Chih-Jung Kuo ; Tzu-Ping Ko ; Min-Feng Hsu ; Yao-Chen Tsui ; Shih-Cheng Chang ; Syaulan Yang ; Shu-Jen Chen ; Hua-Chien Chen ; Ming-Chu Hsu ; Shin-Ru Shih ; Po-Huang Liang ; Andrew H-J Wang | Structural basis of inhibition specificities of 3C and 3C-like proteases by zinc-coordinating and peptidomimetic compounds. |
| 002B97 (2009) |
Krongsakda Phakthanakanok [Thaïlande] ; Khanok Ratanakhanokchai ; Khin Lay Kyu ; Pornthep Sompornpisut ; Aaron Watts ; Surapong Pinitglang | A computational analysis of SARS cysteine proteinase-octapeptide substrate interaction: implication for structure and active site binding mechanism. |
| 003072 (2008) |
Chunying Niu [Canada] ; Jiang Yin ; Jianmin Zhang ; John C. Vederas ; Michael N G. James | Molecular docking identifies the binding of 3-chloropyridine moieties specifically to the S1 pocket of SARS-CoV Mpro. |
| 003584 (2007) |
D H Goetz [États-Unis] ; Y. Choe ; E. Hansell ; Y T Chen ; M. Mcdowell ; C B Jonsson ; W R Roush ; J. Mckerrow ; C S Craik | Substrate specificity profiling and identification of a new class of inhibitor for the major protease of the SARS coronavirus. |
| 004873 (2005) |
Haitao Yang [République populaire de Chine] ; Weiqing Xie ; Xiaoyu Xue ; Kailin Yang ; Jing Ma ; Wenxue Liang ; Qi Zhao ; Zhe Zhou ; Duanqing Pei ; John Ziebuhr ; Rolf Hilgenfeld ; Kwok Yung Yuen ; Luet Wong ; Guangxia Gao ; Saijuan Chen ; Zhu Chen ; Dawei Ma ; Mark Bartlam ; Zihe Rao | Design of wide-spectrum inhibitors targeting coronavirus main proteases. |
| 004923 (2005) |
Qishi Du [République populaire de Chine] ; Shuqing Wang ; Zhiqin Jiang ; Weina Gao ; Yun Li ; Dongqing Wei ; Kuo-Chen Chou | Application of bioinformatics in search for cleavable peptides of SARS-CoV M(pro) and chemical modification of octapeptides. |
| 004973 (2005) |
Yu-San Han [République populaire de Chine] ; Gu-Gang Chang [République populaire de Chine] ; Chiun-Gung Juo [République populaire de Chine] ; Hong-Jen Lee [République populaire de Chine] ; Shiou-Hwei Yeh [République populaire de Chine] ; John Tsu-An Hsu [République populaire de Chine] ; Xin Chen [République populaire de Chine, Taïwan] | Papain-Like Protease 2 (PLP2) from Severe Acute Respiratory Syndrome Coronavirus (SARS-CoV): Expression, Purification, Characterization, and Inhibition† |
