Serveur d'exploration SRAS - Exploration (Accueil)

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0219-3116 < 0223-5234 < 0235-2990  Facettes :

List of bibliographic references indexed by 0223-5234

Number of relevant bibliographic references: 14.
Ident.Authors (with country if any)Title
000B96 (2018-09) Cyril Fersing [France] ; Clotilde Boudot [France] ; Julien Pedron [France] ; Sébastien Hutter [France] ; Nicolas Primas [France] ; Caroline Castera-Ducros [France] ; Sandra Bourgeade-Delmas [France] ; Alix Sournia-Saquet [France] ; Alain Moreau [France] ; Anita Cohen [France] ; Jean-Luc Stigliani [France] ; Geneviève Pratviel [France] ; Maxime Crozet [France] ; Susan Wyllie [Royaume-Uni] ; Alan Fairlamb [Royaume-Uni] ; Alexis Valentin [France] ; Pascal Rathelot [France] ; Nadine Azas [France] ; Bertrand Courtioux [France] ; Pierre Verhaeghe [France] ; Patrice Vanelle [France]8-Aryl-6-chloro-3-nitro-2-(phenylsulfonylmethyl)imidazo[1,2-a]pyridines as potent antitrypanosomatid molecules bioactivated by type 1 nitroreductases
000D34 (2017) Justine Desroches [France] ; Charline Kieffer [France] ; Nicolas Primas [France] ; Sébastien Hutter [France] ; Armand Gellis [France] ; Hussein El-Kashef [Égypte] ; Pascal Rathelot [France] ; Pierre Verhaeghe [France] ; Nadine Azas [France] ; Patrice Vanelle [France]Discovery of new hit-molecules targeting Plasmodium falciparum through a global SAR study of the 4-substituted-2-trichloromethylquinazoline antiplasmodial scaffold
000E50 (2017) Li Wang [République populaire de Chine] ; Bo-Bo Bao [République populaire de Chine] ; Guo-Qing Song [République populaire de Chine] ; Cheng Chen [République populaire de Chine] ; Xu-Meng Zhang [République populaire de Chine] ; Wei Lu [République populaire de Chine] ; Zefang Wang [République populaire de Chine] ; Yan Cai [République populaire de Chine] ; Shuang Li [République populaire de Chine] ; Sheng Fu [République populaire de Chine] ; Fu-Hang Song [République populaire de Chine] ; Haitao Yang [République populaire de Chine] ; Jian-Guo Wang [République populaire de Chine]Discovery of unsymmetrical aromatic disulfides as novel inhibitors of SARS-CoV main protease: Chemical synthesis, biological evaluation, molecular docking and 3D-QSAR study
000F05 (2016) Armand Gellis [France] ; Nicolas Primas [France] ; Sébastien Hutter [France] ; Gilles Lanzada [France] ; Vincent Remusat [France] ; Pierre Verhaeghe [France] ; Patrice Vanelle [France] ; Nadine Azas [France]Looking for new antiplasmodial quinazolines: DMAP-catalyzed synthesis of 4-benzyloxy- and 4-aryloxy-2-trichloromethylquinazolines and their in vitro evaluation toward Plasmodium falciparum
001518 (2014) Nicolas Primas [France] ; Peggy Suzanne [France] ; Pierre Verhaeghe [France] ; Sébastien Hutter [France] ; Charline Kieffer [France] ; Michèle Laget [France] ; Anita Cohen [France] ; Julie Broggi [France] ; Jean-Charles Lancelot [France] ; Aurélien Lesnard [France] ; Patrick Dallemagne [France] ; Pascal Rathelot [France] ; Sylvain Rault [France] ; Patrice Vanelle [France] ; Nadine Azas [France]Synthesis and in vitro evaluation of 4-trichloromethylpyrrolo[1,2-a]quinoxalines as new antiplasmodial agents
001964 (2013) Pillaiyar Thanigaimalai [Japon] ; Sho Konno [Japon] ; Takehito Yamamoto [Japon] ; Yuji Koiwai [Japon] ; Akihiro Taguchi [Japon] ; Kentaro Takayama [Japon] ; Fumika Yakushiji [Japon] ; Kenichi Akaji [Japon] ; Yoshiaki Kiso [Japon] ; Yuko Kawasaki [États-Unis] ; Shen-En Chen [États-Unis] ; Aurash Naser-Tavakolian [États-Unis] ; Arne Schön [États-Unis] ; Ernesto Freire [États-Unis] ; Yoshio Hayashi [Japon]Design, synthesis, and biological evaluation of novel dipeptide-type SARS-CoV 3CL protease inhibitors: Structure–activity relationship study
002357 (2011) Rui-Hua Guo [République populaire de Chine] ; QUAN ZHANG [République populaire de Chine] ; Yun-Bao Ma [République populaire de Chine] ; JIE LUO [République populaire de Chine] ; Chang-An Geng [République populaire de Chine] ; Li-Jun Wang [République populaire de Chine] ; Xue-Mei Zhang [République populaire de Chine] ; JUN ZHOU [République populaire de Chine] ; Zhi-Yong Jiang [République populaire de Chine] ; Ji-Jun Chen [République populaire de Chine]Structure-activity relationships study of 6-chloro-4-(2-chlorophenyl)-3-(2-hydroxyethyl) quinolin-2(1H)-one derivatives as novel non-nucleoside anti-hepatitis B virus agents
002392 (2011) MI KYOUNG KIM [Corée du Sud] ; Mi-Sun Yu [Corée du Sud] ; HYE RI PARKA [Corée du Sud] ; KYUNG BO KIM [Corée du Sud] ; Chaewoon Lee [Corée du Sud] ; SUH YOUNG CHO [Corée du Sud] ; Jihoon Kang [Corée du Sud] ; Hyunjun Yoon [Corée du Sud] ; Dong-Eun Kim [Corée du Sud] ; Hyunah Choo [Corée du Sud] ; Yong-Joo Jeong [Corée du Sud] ; Youhoon Chong [Corée du Sud]2,6-Bis-arylmethyloxy-5-hydroxychromones with antiviral activity against both hepatitis C virus (HCV) and SARS-associated coronavirus (SCV)
002F04 (2009) Yue-Ping Wang [République populaire de Chine] ; Fen-Er Chen [République populaire de Chine] ; Erik De Clercq [Belgique] ; Jan Balzarini [Belgique] ; Christophe Pannecouque [Belgique]Synthesis and in vitro anti-HIV evaluation of a new series of 6-arylmethyl-substituted S-DABOs as potential non-nucleoside HIV-1 reverse transcriptase inhibitors
002F19 (2009) Andrea Spallarossa [Italie] ; Sara Cesarini [Italie] ; Angelo Ranise [Italie] ; Silvia Schenone [Italie] ; Olga Bruno [Italie] ; Alberto Borassi [Italie] ; Paolo La Colla [Italie] ; Margherita Pezzullo [Italie] ; Giuseppina Sanna [Italie] ; Gabriella Collu [Italie] ; Barbara Secci [Italie] ; Roberta Loddo [Italie]Parallel synthesis, molecular modelling and further structure-activity relationship studies of new acylthiocarbamates as potent non-nucleoside HIV-1 reverse transcriptase inhibitors
002F21 (2009) Andrea Spallarossa [Italie] ; Sara Cesarini [Italie] ; Angelo Ranise [Italie] ; Olga Bruno [Italie] ; Silvia Schenone [Italie] ; Paolo La Colla [Italie] ; Gabriella Collu [Italie] ; Giuseppina Sanna [Italie] ; Barbara Secci [Italie] ; Roberta Loddo [Italie]Novel modifications in the series of O-(2-phthalimidoethyl)-N-substituted thiocarbamates and their ring-opened congeners as non-nucleoside HIV-1 reverse transcriptase inhibitors
004409 (2006) Yue-Qing Li [République populaire de Chine] ; Ze-Lin Li [République populaire de Chine] ; Wei-Jie Zhao [République populaire de Chine] ; Rui-Xing Wen [République populaire de Chine] ; Qing-Wei Meng [République populaire de Chine] ; YI ZENG [République populaire de Chine]Synthesis of stilbene derivatives with inhibition of SARS coronavirus replication
004823 (2005) Xue Wu Zhang [Hong Kong] ; Yee Leng Yap ; Ralf M. AltmeyerGeneration of predictive pharmacophore model for SARS-coronavirus main proteinase.
004E22 (2005) XUE WU ZHANG [Hong Kong] ; YEE LENG YAP [Hong Kong] ; Ralf M. Altmeyer [Hong Kong]Generation of predictive pharmacophore model for SARS-coronavirus main proteinase

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