6SLN-lipo PGA specifically catches (coats) human influenza virus and synergizes neuraminidase-targeting drugs for human influenza therapeutic potential.
Identifieur interne : 001A51 ( Ncbi/Curation ); précédent : 001A50; suivant : 001A526SLN-lipo PGA specifically catches (coats) human influenza virus and synergizes neuraminidase-targeting drugs for human influenza therapeutic potential.
Auteurs : Nongluk Sriwilaijaroen [Oman] ; Katsuhiko Suzuki [Japon] ; Emi Takashita [Japon] ; Hiroaki Hiramatsu [Japon] ; Osamu Kanie [Japon] ; Yasuo Suzuki [Japon]Source :
- The Journal of antimicrobial chemotherapy [ 1460-2091 ] ; 2015.
Descripteurs français
- KwdFr :
- Acide polyglutamique (), Acide polyglutamique (analogues et dérivés), Acide polyglutamique (pharmacologie), Acide polyglutamique (synthèse chimique), Animaux, Antienzymes (pharmacologie), Antiviraux (), Antiviraux (pharmacologie), Antiviraux (synthèse chimique), Attachement viral (), Concentration inhibitrice 50, Glycolipides (), Glycolipides (pharmacologie), Glycolipides (synthèse chimique), Humains, Liaison aux protéines, Lignée cellulaire, Protéines virales (antagonistes et inhibiteurs), Relation dose-effet des médicaments, Récepteurs viraux (métabolisme), Sialidase (antagonistes et inhibiteurs), Synergie des médicaments, Virus de la grippe A (), Virus de la grippe A (physiologie), Érythrocytes (), Érythrocytes (virologie).
- MESH :
- analogues et dérivés : Acide polyglutamique.
- antagonistes et inhibiteurs : Protéines virales, Sialidase.
- métabolisme : Récepteurs viraux.
- pharmacologie : Acide polyglutamique, Antienzymes, Antiviraux, Glycolipides.
- physiologie : Virus de la grippe A.
- synthèse chimique : Acide polyglutamique, Antiviraux, Glycolipides.
- virologie : Érythrocytes.
- Acide polyglutamique, Animaux, Antiviraux, Attachement viral, Concentration inhibitrice 50, Glycolipides, Humains, Liaison aux protéines, Lignée cellulaire, Relation dose-effet des médicaments, Synergie des médicaments, Virus de la grippe A, Érythrocytes.
English descriptors
- KwdEn :
- Animals, Antiviral Agents (chemical synthesis), Antiviral Agents (chemistry), Antiviral Agents (pharmacology), Cell Line, Dose-Response Relationship, Drug, Drug Synergism, Enzyme Inhibitors (pharmacology), Erythrocytes (drug effects), Erythrocytes (virology), Glycolipids (chemical synthesis), Glycolipids (chemistry), Glycolipids (pharmacology), Humans, Influenza A virus (drug effects), Influenza A virus (physiology), Inhibitory Concentration 50, Neuraminidase (antagonists & inhibitors), Polyglutamic Acid (analogs & derivatives), Polyglutamic Acid (chemical synthesis), Polyglutamic Acid (chemistry), Polyglutamic Acid (pharmacology), Protein Binding, Receptors, Virus (metabolism), Viral Proteins (antagonists & inhibitors), Virus Attachment (drug effects).
- MESH :
- chemical , analogs & derivatives : Polyglutamic Acid.
- chemical , antagonists & inhibitors : Neuraminidase, Viral Proteins.
- chemical , chemical synthesis : Antiviral Agents, Glycolipids, Polyglutamic Acid.
- chemical , chemistry : Antiviral Agents, Glycolipids, Polyglutamic Acid.
- chemical , metabolism : Receptors, Virus.
- chemical , pharmacology : Antiviral Agents, Enzyme Inhibitors, Glycolipids, Polyglutamic Acid.
- drug effects : Erythrocytes, Influenza A virus, Virus Attachment.
- physiology : Influenza A virus.
- virology : Erythrocytes.
- Animals, Cell Line, Dose-Response Relationship, Drug, Drug Synergism, Humans, Inhibitory Concentration 50, Protein Binding.
Abstract
The purpose of this study was to develop a new compound to overcome influenza epidemics and pandemics as well as drug resistance.
DOI: 10.1093/jac/dkv193
PubMed: 26169554
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pubmed:26169554Le document en format XML
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<affiliation wicri:level="1"><nlm:affiliation>Department of Preclinical Sciences, Faculty of Medicine, Thammasat University (Rangsit Campus), Pathumthani 12120, Thailand College of Life and Health Sciences, Chubu University, Aichi 487-8501, Japan snongluk@hotmail.com.</nlm:affiliation>
<country wicri:rule="url">Oman</country>
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<term>Antiviral Agents (chemical synthesis)</term>
<term>Antiviral Agents (chemistry)</term>
<term>Antiviral Agents (pharmacology)</term>
<term>Cell Line</term>
<term>Dose-Response Relationship, Drug</term>
<term>Drug Synergism</term>
<term>Enzyme Inhibitors (pharmacology)</term>
<term>Erythrocytes (drug effects)</term>
<term>Erythrocytes (virology)</term>
<term>Glycolipids (chemical synthesis)</term>
<term>Glycolipids (chemistry)</term>
<term>Glycolipids (pharmacology)</term>
<term>Humans</term>
<term>Influenza A virus (drug effects)</term>
<term>Influenza A virus (physiology)</term>
<term>Inhibitory Concentration 50</term>
<term>Neuraminidase (antagonists & inhibitors)</term>
<term>Polyglutamic Acid (analogs & derivatives)</term>
<term>Polyglutamic Acid (chemical synthesis)</term>
<term>Polyglutamic Acid (chemistry)</term>
<term>Polyglutamic Acid (pharmacology)</term>
<term>Protein Binding</term>
<term>Receptors, Virus (metabolism)</term>
<term>Viral Proteins (antagonists & inhibitors)</term>
<term>Virus Attachment (drug effects)</term>
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<term>Acide polyglutamique (analogues et dérivés)</term>
<term>Acide polyglutamique (pharmacologie)</term>
<term>Acide polyglutamique (synthèse chimique)</term>
<term>Animaux</term>
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<term>Antiviraux (pharmacologie)</term>
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<term>Concentration inhibitrice 50</term>
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<term>Glycolipides (pharmacologie)</term>
<term>Glycolipides (synthèse chimique)</term>
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<term>Liaison aux protéines</term>
<term>Lignée cellulaire</term>
<term>Protéines virales (antagonistes et inhibiteurs)</term>
<term>Relation dose-effet des médicaments</term>
<term>Récepteurs viraux (métabolisme)</term>
<term>Sialidase (antagonistes et inhibiteurs)</term>
<term>Synergie des médicaments</term>
<term>Virus de la grippe A ()</term>
<term>Virus de la grippe A (physiologie)</term>
<term>Érythrocytes ()</term>
<term>Érythrocytes (virologie)</term>
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<keywords scheme="MESH" type="chemical" qualifier="analogs & derivatives" xml:lang="en"><term>Polyglutamic Acid</term>
</keywords>
<keywords scheme="MESH" type="chemical" qualifier="antagonists & inhibitors" xml:lang="en"><term>Neuraminidase</term>
<term>Viral Proteins</term>
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<keywords scheme="MESH" type="chemical" qualifier="chemical synthesis" xml:lang="en"><term>Antiviral Agents</term>
<term>Glycolipids</term>
<term>Polyglutamic Acid</term>
</keywords>
<keywords scheme="MESH" type="chemical" qualifier="chemistry" xml:lang="en"><term>Antiviral Agents</term>
<term>Glycolipids</term>
<term>Polyglutamic Acid</term>
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<keywords scheme="MESH" type="chemical" qualifier="metabolism" xml:lang="en"><term>Receptors, Virus</term>
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<keywords scheme="MESH" type="chemical" qualifier="pharmacology" xml:lang="en"><term>Antiviral Agents</term>
<term>Enzyme Inhibitors</term>
<term>Glycolipids</term>
<term>Polyglutamic Acid</term>
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<keywords scheme="MESH" qualifier="analogues et dérivés" xml:lang="fr"><term>Acide polyglutamique</term>
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<keywords scheme="MESH" qualifier="antagonistes et inhibiteurs" xml:lang="fr"><term>Protéines virales</term>
<term>Sialidase</term>
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<term>Virus Attachment</term>
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<keywords scheme="MESH" qualifier="pharmacologie" xml:lang="fr"><term>Acide polyglutamique</term>
<term>Antienzymes</term>
<term>Antiviraux</term>
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<keywords scheme="MESH" qualifier="synthèse chimique" xml:lang="fr"><term>Acide polyglutamique</term>
<term>Antiviraux</term>
<term>Glycolipides</term>
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<keywords scheme="MESH" qualifier="virologie" xml:lang="fr"><term>Érythrocytes</term>
</keywords>
<keywords scheme="MESH" qualifier="virology" xml:lang="en"><term>Erythrocytes</term>
</keywords>
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<term>Cell Line</term>
<term>Dose-Response Relationship, Drug</term>
<term>Drug Synergism</term>
<term>Humans</term>
<term>Inhibitory Concentration 50</term>
<term>Protein Binding</term>
</keywords>
<keywords scheme="MESH" xml:lang="fr"><term>Acide polyglutamique</term>
<term>Animaux</term>
<term>Antiviraux</term>
<term>Attachement viral</term>
<term>Concentration inhibitrice 50</term>
<term>Glycolipides</term>
<term>Humains</term>
<term>Liaison aux protéines</term>
<term>Lignée cellulaire</term>
<term>Relation dose-effet des médicaments</term>
<term>Synergie des médicaments</term>
<term>Virus de la grippe A</term>
<term>Érythrocytes</term>
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<front><div type="abstract" xml:lang="en">The purpose of this study was to develop a new compound to overcome influenza epidemics and pandemics as well as drug resistance.</div>
</front>
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