Ident. | Authors (with country if any) | Title |
---|
000072 (2020) |
Shan-Meng Lin [Taïwan] ; Shih-Chao Lin [États-Unis] ; Jia-Ning Hsu [Taïwan] ; Chung-Ke Chang [Taïwan] ; Ching-Ming Chien [Taïwan] ; Yong-Sheng Wang [Taïwan] ; Hung-Yi Wu [Taïwan] ; U-Ser Jeng [Taïwan] ; Kylene Kehn-Hall [États-Unis] ; Ming-Hon Hou [Taïwan] | Structure-Based
Stabilization of Non-native Protein–Protein
Interactions of Coronavirus Nucleocapsid Proteins in Antiviral Drug
Design |
000630 (2019) |
Ji-Seong Yoon [Corée du Sud] ; Gyudong Kim [Corée du Sud] ; Dnyandev B. Jarhad [Corée du Sud] ; Hong-Rae Kim [Corée du Sud] ; Young-Sup Shin [Corée du Sud] ; Shuhao Qu [Corée du Sud, République populaire de Chine] ; Pramod K. Sahu [Corée du Sud] ; Hea Ok Kim [Corée du Sud] ; Hyuk Woo Lee [Corée du Sud] ; Su Bin Wang [Corée du Sud] ; Yun Jeong Kong [Corée du Sud] ; Tong-Shin Chang [Corée du Sud] ; Natacha S. Ogando [Pays-Bas] ; Kristina Kovacikova [Pays-Bas] ; Eric J. Snijder [Pays-Bas] ; Clara C. Posthuma [Pays-Bas] ; Martijn J. Van Hemert [Pays-Bas] ; Lak Shin Jeong [Corée du Sud] | Design, Synthesis,
and Anti-RNA Virus Activity of
6′-Fluorinated-Aristeromycin Analogues |
000A03 (2018) |
Chao Wang [République populaire de Chine] ; Shuai Xia [République populaire de Chine] ; Peiyu Zhang [République populaire de Chine] ; Tianhong Zhang [République populaire de Chine] ; Weicong Wang [République populaire de Chine] ; Yangli Tian [République populaire de Chine] ; Guangpeng Meng [République populaire de Chine] ; Shibo Jiang [République populaire de Chine, États-Unis] ; Keliang Liu [République populaire de Chine] | Discovery of Hydrocarbon-Stapled
Short α-Helical
Peptides as Promising Middle East Respiratory Syndrome Coronavirus
(MERS-CoV) Fusion Inhibitors |
000A15 (2018) |
Chao Wang [République populaire de Chine] ; Lei Zhao [République populaire de Chine] ; Shuai Xia [République populaire de Chine] ; Tianhong Zhang [République populaire de Chine] ; Ruiyuan Cao [République populaire de Chine] ; Guodong Liang [République populaire de Chine] ; Yue Li [République populaire de Chine] ; Guangpeng Meng [République populaire de Chine] ; Weicong Wang [République populaire de Chine] ; Weiguo Shi [République populaire de Chine] ; Wu Zhong [République populaire de Chine] ; Shibo Jiang [République populaire de Chine, États-Unis] ; Keliang Liu [République populaire de Chine] | De Novo Design
of α-Helical Lipopeptides
Targeting Viral Fusion Proteins: A Promising Strategy for Relatively
Broad-Spectrum Antiviral Drug Discovery |
003098 (2004) |
Christoph Pisterer [Allemagne] ; Dan Mihailescu [Allemagne] ; Jeremy C. Smith [Allemagne] ; Jennifer Reed [Allemagne] | A Common Pharmacophoric Footprint for AIDS Vaccine Design |
003248 (2003) |
Robyn M. Hyde [États-Unis] ; Arthur D. Broom [États-Unis] ; Robert W. Buckheit [États-Unis] | Antiviral Amphipathic Oligo- and Polyribonucleotides: Analogue Development and Biological Studies |
003663 (2000) |
Alan D. Borthwick [Royaume-Uni] ; S. Jane Angier [Royaume-Uni] ; Andrew J. Crame [Royaume-Uni] ; Anne M. Exall [Royaume-Uni] ; Terry M. Haley [Royaume-Uni] ; Graham J. Hart [Royaume-Uni] ; Andrew M. Mason [Royaume-Uni] ; Andrew M. K. Pennell [Royaume-Uni] ; Gordon G. Weingarten [Royaume-Uni] | Design and Synthesis of Pyrrolidine-5,5-trans-lactams (5-Oxo-hexahydro-pyrrolo[3,2-b]pyrroles) as Novel Mechanism-Based Inhibitors of Human Cytomegalovirus Protease. 1. The α-Methyl-trans-lactam Template |
003A31 (1998) |
Bernd Eschgf Ller [Suisse] ; Marcel König [Suisse] ; Franziska Boess [Suisse] ; Urs A. Boelsterli [Suisse] ; Steven A. Benner [Suisse] | Synthesis and Biodistribution of a Short Nonionic Oligonucleotide Analogue in Mouse with a Potential to Mimic Peptides |
003A90 (1998) |
Hitoshi Hotoda [Japon] ; Makoto Koizumi [Japon] ; Rika Koga [Japon] ; Masakatsu Kaneko [Japon] ; Kenji Momota [Japon] ; Toshinori Ohmine [Japon] ; Hidehiko Furukawa [Japon] ; Toshinori Agatsuma [Japon] ; Takashi Nishigaki [Japon] ; Junko Sone [Japon] ; Shinya Tsutsumi [Japon] ; Toshiyuki Kosaka [Japon] ; Koji Abe [Japon] ; Satoshi Kimura [Japon] ; Kaoru Shimada [Japon] | Biologically Active Oligodeoxyribonucleotides. 5. 5‘-End-Substituted d(TGGGAG) Possesses Anti-Human Immunodeficiency Virus Type 1 Activity by Forming a G-Quadruplex Structure |
003E30 (1996) |
M M Javadpour [États-Unis] ; M M Juban ; W C Lo ; S M Bishop ; J B Alberty ; S M Cowell ; C L Becker ; M L Mclaughlin | De novo antimicrobial peptides with low mammalian cell toxicity. |
003E95 (1996) |
Danielle A. M. Konings [États-Unis] ; Jacqueline R. Wyatt [États-Unis] ; David J. Ecker [États-Unis] ; Susan M. Freier [États-Unis] | Deconvolution of Combinatorial Libraries for Drug Discovery: Theoretical Comparison of Pooling Strategies |
004004 (1995-10-01) |
Michael W. Reed ; Eugeny Lukhtanov ; Vladimir Gorn ; Deborah D. Lucas ; James H. Zhou ; S. Balakrishna Pai ; Yung-Chi Cheng ; Rich B. Meyer | Structure-Activity Relationships of Cytotoxic Cholesterol-Modified DNA Duplexes |
004005 (1995-10-01) |
Mathai Mammen ; Georg Dahmann ; George M. Whitesides | Effective Inhibitors of Hemagglutination by Influenza Virus Synthesized from Polymers Having Active Ester Groups. Insight into Mechanism of Inhibition |
004014 (1995-01-01) |
Susan M. Freier ; Danielle A. M. Konings ; Jacqueline R. Wyatt ; David J. Ecker | Deconvolution of Combinatorial Libraries for Drug Discovery: A Model System |
004043 (1995) |
D S Jones [États-Unis] ; P A Barstad ; M J Feild ; J P Hachmann ; M S Hayag ; K W Hill ; G M Iverson ; D A Livingston ; M S Palanki ; A R Tibbetts | Immunospecific reduction of antioligonucleotide antibody-forming cells with a tetrakis-oligonucleotide conjugate (LJP 394), a therapeutic candidate for the treatment of lupus nephritis. |
004247 (1994-05-01) |
Eric M. Gordon ; Ronald W. Barrett ; William J. Dower ; Stephen P. A. Fodor ; Mark A. Gallop | Applications of Combinatorial Technologies to Drug Discovery. 2. Combinatorial Organic Synthesis, Library Screening Strategies, and Future Directions |
004494 (1993-07-01) |
John F. Milligan ; Mark D. Matteucci ; John C. Martin | Current concepts in antisense drug design |
004706 (1992-08-01) |
Jeh Jeng Wang ; G. Craig Hill ; Laurence H. Hurley | Template-directed design of a DNA-DNA crosslinker based upon a bis-tomaymycin-duplex adduct |
004F62 (1980-01-01) |
Wayne K. Anderson ; George E. Lee | Synthesis of 8-methoxy-15,16-dinor-6,8,10-trichothecatriene 12,13.alpha.-epoxide and 12,13.beta.-epoxide as potential antineoplastic agents |
005127 (1973-03-01) |
Arthur D. Sill ; William L. Albrecht ; Edwin R. Andrews ; Robert W. Fleming ; Stephen W. Horgan ; Edward Mcc. Roberts ; F. William Sweet | Bis-basic-substituted polycyclic aromatic compounds. New class of antiviral agents. 1. Bisalkamine esters of fluorenone-, fluorenol-, and fluorenedicarboxylic acids |
005168 (1971-06-01) |
Charles G. Skinner ; John D. Huddle | Synthesis of 1-amino-2-hydroxycyclopentanecarboxylic acid |