Eléments de l'association
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List of bibliographic references
Number of relevant bibliographic references: 12.Ident. | Authors (with country if any) | Title |
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000635 | Jozlyn R. Clasman [États-Unis] ; Renata K. Everett [États-Unis] ; Karthik Srinivasan [États-Unis] ; Andrew D. Mesecar [États-Unis] | Decoupling deISGylating and deubiquitinating activities of the MERS virus papain-like protease |
000B18 | Jozlyn R. Clasman [États-Unis] ; Yahira M. Báez-Santos [États-Unis] ; Robert C. Mettelman [États-Unis] ; Amornrat O Rien [États-Unis] ; Susan C. Baker [États-Unis] ; Andrew D. Mesecar [États-Unis] | X-ray Structure and Enzymatic Activity Profile of a Core Papain-like Protease of MERS Coronavirus with utility for structure-based drug design |
000B77 | Courtney M. Daczkowski [États-Unis] ; John V. Dzimianski [États-Unis] ; Jozlyn R. Clasman [États-Unis] ; Octavia Goodwin [États-Unis] ; Andrew D. Mesecar [États-Unis] ; Scott D. Pegan [États-Unis] | Structural Insights into the Interaction of Coronavirus Papain-Like Proteases and Interferon-Stimulated Gene Product 15 from Different Species |
000E50 | Areej Abuhammad [Jordanie] ; Rua'A A. Al-Aqtash [Jordanie] ; Brandon J. Anson [États-Unis] ; Andrew D. Mesecar [États-Unis] ; Mutasem O. Taha [Jordanie] | Computational modeling of the bat HKU4 coronavirus 3CLpro inhibitors as a tool for the development of antivirals against the emerging Middle East respiratory syndrome (MERS) coronavirus. |
001553 | Sarah E. St. John [États-Unis] ; Sakshi Tomar [États-Unis] ; Shaun R. Stauffer [États-Unis] ; Andrew D. Mesecar [États-Unis] | Targeting zoonotic viruses: Structure-based inhibition of the 3C-like protease from bat coronavirus HKU4—The likely reservoir host to the human coronavirus that causes Middle East Respiratory Syndrome (MERS) |
001719 | Sakshi Tomar ; Melanie L. Johnston [États-Unis] ; Sarah E. St. John ; Heather L. Osswald [États-Unis] ; Prasanth R. Nyalapatla [États-Unis] ; Lake N. Paul ; Arun K. Ghosh [États-Unis] ; Mark R. Denison ; Andrew D. Mesecar [États-Unis] | Ligand-induced Dimerization of Middle East Respiratory Syndrome (MERS) Coronavirus nsp5 Protease (3CLpro) |
001B31 | Anna M. Mielech [États-Unis] ; Yafang Chen [États-Unis] ; Andrew D. Mesecar [États-Unis] ; Susan C. Baker [États-Unis] | Nidovirus papain-like proteases: multifunctional enzymes with protease, deubiquitinating and deISGylating activities. |
001D05 | Xufang Deng [États-Unis] ; Sarah E. Stjohn [États-Unis] ; Heather L. Osswald [États-Unis] ; Amornrat O'Brien [États-Unis] ; Bridget S. Banach [États-Unis] ; Katrina Sleeman [États-Unis] ; Arun K. Ghosh [États-Unis] ; Andrew D. Mesecar [États-Unis] ; Susan C. Baker [États-Unis] | Coronaviruses resistant to a 3C-like protease inhibitor are attenuated for replication and pathogenesis, revealing a low genetic barrier but high fitness cost of resistance. |
001D24 | Yahira M. Báez-Santos [États-Unis] ; Anna M. Mielech [États-Unis] ; Xufang Deng [États-Unis] ; Susan Baker [États-Unis] ; Andrew D. Mesecar [États-Unis] | Catalytic function and substrate specificity of the papain-like protease domain of nsp3 from the Middle East respiratory syndrome coronavirus. |
001D63 | Xufang Deng [États-Unis] ; Sudhakar Agnihothram [États-Unis] ; Anna M. Mielech [États-Unis] ; Daniel B. Nichols [États-Unis] ; Michael W. Wilson [États-Unis] ; Sarah E. Stjohn [États-Unis] ; Scott D. Larsen [États-Unis] ; Andrew D. Mesecar [États-Unis] ; Deborah J. Lenschow [États-Unis] ; Ralph S. Baric [États-Unis] ; Susan C. Baker [États-Unis] | A chimeric virus-mouse model system for evaluating the function and inhibition of papain-like proteases of emerging coronaviruses. |
001F63 | Anna M. Mielech [États-Unis] ; Andy Kilianski [États-Unis] ; Yahira M. Baez-Santos [États-Unis] ; Andrew D. Mesecar [États-Unis] ; Susan C. Baker [États-Unis] | MERS-CoV papain-like protease has deISGylating and deubiquitinating activities |
002011 | Mark Turlington [États-Unis] ; Aspen Chun ; Sakshi Tomar ; Aimee Eggler ; Valerie Grum-Tokars ; Jon Jacobs ; J Scott Daniels ; Eric Dawson ; Adrian Saldanha ; Peter Chase ; Yahira M. Baez-Santos ; Craig W. Lindsley ; Peter Hodder ; Andrew D. Mesecar ; Shaun R. Stauffer | Discovery of N-(benzo[1,2,3]triazol-1-yl)-N-(benzyl)acetamido)phenyl) carboxamides as severe acute respiratory syndrome coronavirus (SARS-CoV) 3CLpro inhibitors: identification of ML300 and noncovalent nanomolar inhibitors with an induced-fit binding. |
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