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Poly(2‐oxazoline)s as Polymer Therapeutics

Identifieur interne : 002793 ( Istex/Corpus ); précédent : 002792; suivant : 002794

Poly(2‐oxazoline)s as Polymer Therapeutics

Auteurs : Robert Luxenhofer ; Yingchao Han ; Anita Schulz ; Jing Tong ; Zhijian He ; Alexander V. Kabanov ; Rainer Jordan

Source :

RBID : ISTEX:5E1BC39352B17B4BD0149DD62712F01324AD6FBB

English descriptors

Abstract

Poly(2‐oxazoline)s (POx) are currently discussed as an upcoming polymer platform for biomaterials design and especially for polymer therapeutics. POx meet specific requirements needed for the development of next‐generation polymer therapeutics such as biocompatibility, high modulation of solubility, variation of size, architecture as well as chemical functionality. Although in the early 1990s first and promising POx‐based systems were presented, the field lay dormant for almost two decades. Only very recently, POx‐based polymer therapeutics came back into the focus of very intensive research. In this review, we give an overview on the chemistry and physicochemical properties of POx and summarize the research of POx–protein conjugates, POx–drug conjugates, POx‐based polyplexes and POx micelles for drug delivery.
Poly(2‐oxazoline) (POx) is currently discussed as the upcoming polymer platform for biomaterials design and especially for the development of next‐generation polymer therapeutics. In this review, we give an overview on the chemistry and properties of POx and summarize the research on POx–protein conjugates, POx–drug conjugates, POx‐based polyplexes, and POx micelles for drug delivery.

Url:
DOI: 10.1002/marc.201200354

Links to Exploration step

ISTEX:5E1BC39352B17B4BD0149DD62712F01324AD6FBB

Le document en format XML

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<div type="abstract" xml:lang="en">Poly(2‐oxazoline)s (POx) are currently discussed as an upcoming polymer platform for biomaterials design and especially for polymer therapeutics. POx meet specific requirements needed for the development of next‐generation polymer therapeutics such as biocompatibility, high modulation of solubility, variation of size, architecture as well as chemical functionality. Although in the early 1990s first and promising POx‐based systems were presented, the field lay dormant for almost two decades. Only very recently, POx‐based polymer therapeutics came back into the focus of very intensive research. In this review, we give an overview on the chemistry and physicochemical properties of POx and summarize the research of POx–protein conjugates, POx–drug conjugates, POx‐based polyplexes and POx micelles for drug delivery.</div>
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<json:string>Lai</json:string>
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<json:string>D. W. Kim</json:string>
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<p>Poly(2‐oxazoline)s (POx) are currently discussed as an upcoming polymer platform for biomaterials design and especially for polymer therapeutics. POx meet specific requirements needed for the development of next‐generation polymer therapeutics such as biocompatibility, high modulation of solubility, variation of size, architecture as well as chemical functionality. Although in the early 1990s first and promising POx‐based systems were presented, the field lay dormant for almost two decades. Only very recently, POx‐based polymer therapeutics came back into the focus of very intensive research. In this review, we give an overview on the chemistry and physicochemical properties of POx and summarize the research of POx–protein conjugates, POx–drug conjugates, POx‐based polyplexes and POx micelles for drug delivery.</p>
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<p>Poly(2‐oxazoline)s (POx) are currently discussed as an upcoming polymer platform for biomaterials design and especially for polymer therapeutics. POx meet specific requirements needed for the development of next‐generation polymer therapeutics such as biocompatibility, high modulation of solubility, variation of size, architecture as well as chemical functionality. Although in the early 1990s first and promising POx‐based systems were presented, the field lay dormant for almost two decades. Only very recently, POx‐based polymer therapeutics came back into the focus of very intensive research. In this review, we give an overview on the chemistry and physicochemical properties of POx and summarize the research of POx–protein conjugates, POx–drug conjugates, POx‐based polyplexes and POx micelles for drug delivery.</p>
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<b>Poly(2‐oxazoline) (POx) is currently discussed as the upcoming</b>
polymer platform for biomaterials design and especially for the development of next‐generation polymer therapeutics. In this review, we give an overview on the chemistry and properties of POx and summarize the research on POx–protein conjugates, POx–drug conjugates, POx‐based polyplexes, and POx micelles for drug delivery.
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<title>Poly(2‐oxazoline)s as Polymer Therapeutics</title>
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<name type="personal">
<namePart type="given">Robert</namePart>
<namePart type="family">Luxenhofer</namePart>
<affiliation>Professur für Makromolekulare Chemie, Department Chemie, Technische Universität Dresden, Zellescher Weg 19, 01069 Dresden, Germany</affiliation>
<affiliation>E-mail: Robert.Luxenhofer@chemie.tu‐dresden.de</affiliation>
<affiliation>Correspondence address: Professur für Makromolekulare Chemie, Department Chemie, Technische Universität Dresden, Zellescher Weg 19, 01069 Dresden, Germany.</affiliation>
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<namePart type="given">Yingchao</namePart>
<namePart type="family">Han</namePart>
<affiliation>Center for Drug Delivery and Nanomedicine and Department of Pharmaceutical Sciences, College of Pharmacy, University of Nebraska Medical Center, Omaha, NE 68198‐5830, USA</affiliation>
<affiliation>Biomedical Materials and Engineering Center, Wuhan University of Technology, Wuhan 430070, P. R. China</affiliation>
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<namePart type="given">Anita</namePart>
<namePart type="family">Schulz</namePart>
<affiliation>Professur für Makromolekulare Chemie, Department Chemie, Technische Universität Dresden, Zellescher Weg 19, 01069 Dresden, Germany</affiliation>
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<namePart type="given">Jing</namePart>
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<affiliation>Center for Drug Delivery and Nanomedicine and Department of Pharmaceutical Sciences, College of Pharmacy, University of Nebraska Medical Center, Omaha, NE 68198‐5830, USA</affiliation>
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<namePart type="given">Zhijian</namePart>
<namePart type="family">He</namePart>
<affiliation>Center for Drug Delivery and Nanomedicine and Department of Pharmaceutical Sciences, College of Pharmacy, University of Nebraska Medical Center, Omaha, NE 68198‐5830, USA</affiliation>
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<namePart type="given">Alexander V.</namePart>
<namePart type="family">Kabanov</namePart>
<affiliation>Center for Drug Delivery and Nanomedicine and Department of Pharmaceutical Sciences, College of Pharmacy, University of Nebraska Medical Center, Omaha, NE 68198‐5830, USA</affiliation>
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<namePart type="given">Rainer</namePart>
<namePart type="family">Jordan</namePart>
<affiliation>Professur für Makromolekulare Chemie, Department Chemie, Technische Universität Dresden, Zellescher Weg 19, 01069 Dresden, Germany</affiliation>
<affiliation>Center for Regenerative Therapies Dresden (CRTD), Fetscherstr. 105, 01307 Dresden, Germany</affiliation>
<affiliation>E-mail: Rainer.Jordan@tu‐dresden.de</affiliation>
<affiliation>Correspondence address: Professur für Makromolekulare Chemie, Department Chemie, Technische Universität Dresden, Zellescher Weg 19, 01069 Dresden, Germany.</affiliation>
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<abstract lang="en">Poly(2‐oxazoline)s (POx) are currently discussed as an upcoming polymer platform for biomaterials design and especially for polymer therapeutics. POx meet specific requirements needed for the development of next‐generation polymer therapeutics such as biocompatibility, high modulation of solubility, variation of size, architecture as well as chemical functionality. Although in the early 1990s first and promising POx‐based systems were presented, the field lay dormant for almost two decades. Only very recently, POx‐based polymer therapeutics came back into the focus of very intensive research. In this review, we give an overview on the chemistry and physicochemical properties of POx and summarize the research of POx–protein conjugates, POx–drug conjugates, POx‐based polyplexes and POx micelles for drug delivery.</abstract>
<abstract type="graphical" lang="en">Poly(2‐oxazoline) (POx) is currently discussed as the upcoming polymer platform for biomaterials design and especially for the development of next‐generation polymer therapeutics. In this review, we give an overview on the chemistry and properties of POx and summarize the research on POx–protein conjugates, POx–drug conjugates, POx‐based polyplexes, and POx micelles for drug delivery.</abstract>
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<topic>biomaterial</topic>
<topic>cancer</topic>
<topic>drug delivery</topic>
<topic>gene delivery</topic>
<topic>nanomedicine</topic>
<topic>polymer‐conjugates</topic>
<topic>polymer therapeutic</topic>
<topic>polyoxazoline</topic>
<topic>protein</topic>
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