001011 (2016) |
Iwona E. Głowacka [Pologne] ; Dorota G. Piotrowska [Pologne] ; Graciela Andrei [Belgique] ; Dominique Schols [Belgique] ; Robert Snoeck [Belgique] ; Andrzej E. Wr Blewski [Pologne] | Acyclic nucleoside phosphonates containing the amide bond |
000F43 (2016) |
Iwona E. Głowacka ; Rafał Gulej ; Piotr Grzonkowski ; Graciela Andrei ; Dominique Schols ; Robert Snoeck ; Dorota G. Piotrowska | Synthesis and the Biological Activity of Phosphonylated 1,2,3-Triazolenaphthalimide Conjugates |
001055 (2015) |
Iwona E. Głowacka ; Graciela Andrei ; Dominique Schols ; Robert Snoeck ; Dorota G. Piotrowska | Phosphonylated Acyclic Guanosine Analogues with the 1,2,3-Triazole Linker |
000E11 (2018) |
Magdalena Grabkowska-Dru Yc ; Graciela Andrei ; Dominique Schols ; Robert Snoeck ; Dorota G. Piotrowska | Isoxazolidine Conjugates of N3-Substituted 6-Bromoquinazolinones—Synthesis, Anti-Varizella-Zoster Virus, and Anti-Cytomegalovirus Activity |
000F41 (2016) |
Dorota Rygielska-Tokarska [Pologne] ; Graciela Andrei [Belgique] ; Dominique Schols [Belgique] ; Robert Snoeck [Belgique] ; Iwona E. Głowacka [Pologne] | Synthesis, antiviral, cytotoxic and cytostatic evaluation of N1-(phosphonoalkyl)uracil derivatives |
000F62 (2016) |
Dorota G. Piotrowska ; Graciela Andrei ; Dominique Schols ; Robert Snoeck ; Magdalena Grabkowska-Dru Yc | New Isoxazolidine-Conjugates of Quinazolinones—Synthesis, Antiviral and Cytostatic Activity |
001028 (2016) |
Abdelaaziz Ouahrouch [Maroc, Allemagne] ; Moha Taourirte [Maroc] ; Dominique Schols [Belgique] ; Robert Snoeck [Belgique] ; Graciela Andrei [Belgique] ; Joachim W. Engels [Allemagne] ; Hassan B. Lazrek [Maroc] | Design, Synthesis, and Antiviral Activity of Novel Ribonucleosides of 1,2,3‐Triazolylbenzyl‐aminophosphonates |
001177 (2014) |
Emilia Bankowska [Pologne] ; Jan Balzarini [Belgique] ; Iwona E. Głowacka [Pologne] ; Andrzej E. Wr Blewski [Pologne] | Design, synthesis, antiviral and cytotoxic evaluation of novel acyclic phosphonate nucleotide analogues with a 5,6-dihydro-1H-[1,2,3]triazolo[4,5-d]pyridazine-4,7-dione system |
001197 (2014) |
Iwona E. Głowacka [Pologne] ; Jan Balzarini [Belgique] ; Andrzej E. Wr Blewski [Pologne] | Novel Acyclic Phosphonylated 1,2,3‐Triazolonucleosides with an Acetamidomethyl Linker: Synthesis and Biological Activity |
001209 (2014) |
Iwona E. Głowacka [Pologne] ; Jan Balzarini [Belgique] ; Dorota G. Piotrowska [Pologne] | 1‐Amino‐3‐(1H‐1,2,3‐triazol‐1‐yl)propylphosphonates as Acyclic Analogs of Nucleotides |
001272 (2013) |
Iwona E. Głowacka [Pologne] ; Jan Balzarini [Belgique] ; Andrzej E. Wr Blewski [Pologne] | Synthesis of a New Series of Phosphonylated 1,2,3‐Triazoles as Acyclic Analogs of Ribavirin |
001273 (2013) |
Iwona E. Głowacka [Pologne] ; Jan Balzarini [Belgique] ; Andrzej E. Wr Blewski [Pologne] | Synthesis and Biological Evaluation of Novel 1,2,3‐Triazolonucleotides |
001299 (2012) |
Mahesh K. Lakshman [États-Unis] ; Amit Kumar [États-Unis] ; Raghavan Balachandran [États-Unis] ; Billy W. Day [États-Unis] ; Graciela Andrei [Belgique] ; Robert Snoeck [Belgique] ; Jan Balzarini [Belgique] | Synthesis and Biological Properties of C-2 Triazolylinosine Derivatives |
000D75 (2018) |
Ond Ej Baszczy Ski [République tchèque] ; Martin Maxmilian Kaiser [République tchèque] ; Michal Esnek [République tchèque] ; Petra B Ehová [République tchèque] ; Petr Jansa [République tchèque] ; Eliška Procházková [République tchèque] ; Martin Dra Nsk [République tchèque] ; Robert Snoeck [Belgique] ; Graciela Andrei [Belgique] ; Zlatko Janeba [République tchèque] | Xanthine-based acyclic nucleoside phosphonates with potent antiviral activity against varicella-zoster virus and human cytomegalovirus |
001203 (2014) |
Magdalena Łysakowska [Pologne] ; Jan Balzarini [Belgique] ; Dorota G. Piotrowska [Pologne] | Design, Synthesis, Antiviral, and Cytostatic Evaluation of Novel Isoxazolidine Analogs of Homonucleotides |
001223 (2013) |
Kiran Gangarapu [Inde] ; Sarangapani Manda ; Anvesh Jallapally ; Sreekanth Thota [États-Unis] ; Subhas S. Karki ; Jan Balzarini [Belgique] ; Erik De Clercq [Belgique] ; Harukuni Tokuda [Japon] | Synthesis of thiocarbohydrazide and carbohydrazide derivatives as possible biologically active agents |
001346 (2012) |
Subhas S. Karki [Inde] ; Amol A. Kulkarni [Inde] ; Sujeet Kumar [Inde] ; Suresh Kumar Veliyath [Inde] ; Erik De Clercq [Belgique] ; Jan Balzarini [Belgique] | Synthesis and biological evaluation of 2-(5-substituted-1-((diethylamino)methyl)-2-oxoindolin-3-ylidene)- N -substituted-hydrazinecarbothioamides |
001411 (2011) |
Davorka Završnik ; Samija Muratovi ; Damjan Makuc [Slovénie] ; Janez Plavec [Slovénie] ; Mario Cetina [Croatie] ; Ante Nagl [Croatie] ; Erik De Clercq [Belgique] ; Jan Balzarini [Belgique] ; Mladen Mintas [Croatie] | Benzylidene-bis-(4-Hydroxycoumarin) and Benzopyrano-Coumarin Derivatives: Synthesis, 1H/13C-NMR Conformational and X-ray Crystal Structure Studies and In Vitro Antiviral Activity Evaluations |
001613 (2008) |
Ivana Perkovi [Croatie] ; Ivan Butula [Croatie] ; Branka Zorc [Croatie] ; Karlo Hock [Croatie] ; Sandra Kraljevi Paveli [Croatie] ; Krešimir Paveli [Croatie] ; Erik De Clercq [Belgique] ; Jan Balzarini [Belgique] ; Mladen Mintas [Croatie] | Novel Lipophilic Hydroxyurea Derivatives: Synthesis, Cytostatic and Antiviral Activity Evaluations |
000222 (2020) |
Guangdi Li ; Erik De Clercq | Therapeutic options for the 2019 novel coronavirus (2019-nCoV). |
000D30 (2019) |
Ana C. S. Gondim [Brésil] ; Suzete Roberta Da Silva [Brésil] ; Leen Mathys ; Sam Noppen ; Sandra Liekens ; Alexandre Holanda Sampaio [Brésil] ; Celso S. Nagano [Brésil] ; Cintia Renata Costa Rocha [Brésil] ; Kyria S. Nascimento ; Benildo S. Cavada ; Peter J. Sadler ; Jan Balzarini | Potent antiviral activity of carbohydrate-specific algal and leguminous lectins from the Brazilian biodiversity††Electronic supplementary information (ESI) available. See DOI: 10.1039/c8md00508g |
000D32 (2019) |
Belén Martínez-Gualda [Espagne] ; Liang Sun [Belgique] ; Olaia Martí-Marí [Espagne] ; Carmen Mirabelli [Belgique] ; Leen Delang [Belgique] ; Johan Neyts [Belgique] ; Dominique Schols [Belgique] ; María-José Camarasa [Espagne] ; Ana San-Félix [Espagne] | Modifications in the branched arms of a class of dual inhibitors of HIV and EV71 replication expand their antiviral spectrum. |
000F42 (2016) |
Vanessa Parmenopoulou [Grèce] ; Stella Manta [Grèce] ; Athina Dimopoulou [Grèce] ; Nikolaos Kollatos [Grèce] ; Dominique Schols [Belgique] ; Dimitri Komiotis [Grèce] | Synthesis of novel N-acyl-β-d-glucopyranosylamines and ureas as potential lead cytostatic agents |
001020 (2016) |
Eyüp Ba Aran [Turquie] ; Ay Egül Karaküçük-Iyido An [Turquie] ; Dominique Schols [Belgique] ; Emine Elçin Oruç-Emre [Turquie] | Synthesis of Novel Chiral Sulfonamide‐Bearing 1,2,4‐Triazole‐3‐thione Analogs Derived from D‐ and L‐Phenylalanine Esters as Potential Anti‐Influenza Agents |
001254 (2013) |
Christopher Mcguigan [Royaume-Uni] ; Claire Bourdin [Royaume-Uni] ; Marco Derudas [Royaume-Uni] ; Nadège Hamon [Royaume-Uni] ; Karen Hinsinger [Royaume-Uni] ; Sahar Kandil [Royaume-Uni] ; Karolina Madela [Royaume-Uni] ; Silvia Meneghesso [Royaume-Uni] ; Fabrizio Pertusati [Royaume-Uni] ; Michaela Serpi [Royaume-Uni] ; Magdalena Slusarczyk [Royaume-Uni] ; Stanley Chamberlain [États-Unis] ; Alexander Kolykhalov [États-Unis] ; John Vernachio [États-Unis] ; Christophe Vanpouille [États-Unis] ; Andrea Introini [États-Unis] ; Leonid Margolis [États-Unis] ; Jan Balzarini [Belgique] | Design, synthesis and biological evaluation of phosphorodiamidate prodrugs of antiviral and anticancer nucleosides |
001271 (2013) |
Rosa Miralles-Llumà [Espagne] ; Antoni Figueras [Espagne] ; Félix Busqué [Espagne] ; Angel Alvarez-Larena [Espagne] ; Jan Balzarini [Belgique] ; Marta Figueredo [Espagne] ; Josep Font [Espagne] ; Ramon Alibés [Espagne, Canada] ; Jean-Didier Maréchal [Espagne, Canada] | Synthesis, Antiviral Evaluation, and Computational Studies of Cyclobutane and Cyclobutene L‐Nucleoside Analogues |
001274 (2013) |
Esra Tatar [Turquie] ; Lkay Küçükgüzel [Turquie] ; Dirk Daelemans [Belgique] ; Tanaji T. Talele [États-Unis] ; Neerja Kaushik-Basu [États-Unis] ; Erik De Clercq [Belgique] ; Christophe Pannecouque [Belgique] | Some Hydrazones of 2‐Aroylamino‐3‐methylbutanohydrazide: Synthesis, Molecular Modeling Studies, and Identification as Stereoselective Inhibitors of HIV‐1 |
001352 (2012) |
Pradeep Kumar [Inde] ; Balasubramanian Narasimhan [Inde] ; Kalavathy Ramasamy [Malaisie] ; Vasudevan Mani [Malaisie] ; Rakesh Kumar Mishra [Malaisie] ; Abu Bakar Abdul Majeed [Malaisie] ; Erik De Clercq [Belgique] | N ′-[4-[(Substituted imino)methyl]benzylidene]-substituted benzohydrazides: synthesis, antimicrobial, antiviral, and anticancer evaluation, and QSAR studies |
001372 (2011) |
Kazuhiro Haraguchi [Japon] ; Hisashi Shimada [Japon] ; Keigo Kimura [Japon] ; Genta Akutsu [Japon] ; Hiromichi Tanaka [Japon] ; Hiroshi Abe [Japon] ; Takayuki Hamasaki [Japon] ; Masanori Baba [Japon] ; Elizabeth A. Gullen [États-Unis] ; Ginger E. Dutschman [États-Unis] ; Yung-Chi Cheng [États-Unis] ; Jan Balzarini [Belgique] | Synthesis of 4′-Ethynyl-2′-deoxy-4′-thioribonucleosides and Discovery of a Highly Potent and Less Toxic NRTI |
001403 (2011) |
Lawrence P. Tardibono [États-Unis] ; Marvin J. Miller [États-Unis] ; Jan Balzarini [Belgique] | Enantioselective syntheses of carbocyclic nuleosides 5′-homocarbovir, epi-4′-homocarbovir and their cyclopropylamine analogs using facially selective Pd-mediated allylations |
001415 (2011) |
Alamelu Mahalingam [États-Unis] ; Anthony R. Geonnotti [États-Unis] ; Jan Balzarini [Belgique] ; Patrick F. Kiser [États-Unis] | Activity and Safety of Synthetic Lectins Based on Benzoboroxole-Functionalized Polymers for Inhibition of HIV Entry |
001454 (2010) |
Krishnan Suresh Kumar [Inde] ; Swastika Ganguly ; Ravichandran Veerasamy ; Erik De Clercq | Synthesis, antiviral activity and cytotoxicity evaluation of Schiff bases of some 2-phenyl quinazoline-4(3)H-ones. |
001502 (2010) |
KRISHNAN SURESH KUMAR [Inde] ; Swastika Ganguly [Inde] ; Ravichandran Veerasamy [Malaisie] ; Erik De Clercq [Belgique] | Synthesis, antiviral activity and cytotoxicity evaluation of Schiff bases of some 2-phenyl quinazoline-4(3)H-ones |
001599 (2008) |
Pelayo Camps [Belgique, Espagne] ; Ta Nia Go Mez [Belgique, Espagne] ; Diego Mun Oz-Torrero [Belgique, Espagne] ; Jordi Rull [Belgique, Espagne] ; Laura Sa Nchez [Belgique, Espagne] ; Francesca Boschi [Belgique, Espagne] ; Mauro Comes-Franchini [Belgique] ; Alfredo Ricci [Belgique] ; Teresa Calvet [Belgique, Espagne] ; Merce Font-Bardia [Belgique, Espagne] ; Erik De Clercq [Belgique] ; Lieve Naesens [Belgique] | Synthesis and Absolute Configuration of Novel N,O-Psiconucleosides Using (R)-N-Phenylpantolactam as a Resolution Agent |
001648 (2007) |
Isabel Pérez-Castro [Espagne] ; Olga Caama O [Espagne] ; Franco Fernández [Espagne] ; Marcos D. García [Espagne] ; Carmen L Pez [Espagne] ; Erik De Clercq [Belgique] | Synthesis of 4-substituted-1,2,3-triazole carbanucleoside analogues of ribavirin via click chemistry |
001701 (2006) |
Christophe Biot [Belgique, France] ; Wassim Daher [Belgique] ; Natascha Chavain [Belgique] ; Thierry Fandeur [Belgique] ; Jamal Khalife [Belgique] ; Daniel Dive [Belgique] ; Erik De Clercq [Belgique] | Design and Synthesis of Hydroxyferroquine Derivatives with Antimalarial and Antiviral Activities |