Ident. | Authors (with country if any) | Title |
---|
000068 (2019) |
David Pierrot [France] ; Véronique Sinou [France] ; Sok-Siya Bun [France] ; Daniel Parzy [France] ; Nicolas Taudon [France] ; Jean Rodriguez [France] ; Evelyne Ollivier [France] ; Damien Bonne [France] | Design and synthesis of simplified speciophylline analogues and β-carbolines as active molecules against Plasmodium falciparum |
000076 (2018-01-17) |
Jean Guillon [France] ; Anita Cohen [France] ; Rabindra Nath Das [France] ; Clotilde Boudot [France] ; Nassima Meriem Gueddouda [France] ; Stéphane Moreau [France] ; Luisa Ronga [France] ; Solène Savrimoutou [France] ; Louise Basmaciyan [France] ; Camille Tisnerat [France] ; Sacha Mestanier [France] ; Sandra Rubio [France] ; Sophia Amaziane [France] ; Alexandra Dassonville-Klimpt [France] ; Nadine Azas [France] ; Bertrand Courtioux [France] ; Jean-Louis Mergny [France] ; Catherine Mullié ; Pascal Sonnet | Design, synthesis, and antiprotozoal evaluation of new 2,9-bis[(substituted-aminomethyl)phenyl]-1,10-phenanthroline derivatives |
000083 (2018) |
Aliasghar Jarrahpour ; Malihe Aye ; Javad Ameri Rad ; Saeed Yousefinejad [Iran] ; Veronique Sinou [France] ; Christine Latour [France] ; Jean Michel Brunel [France] ; Edward Turos | Design, synthesis, activity evaluation and QSAR studies of novel antimalarial 1,2,3-triazolo-beta-lactam derivatives |
000099 (2017-05) |
Aida Chaker [France] ; Ennaji Najahi [France] ; Olivier Chatriant [France] ; Alexis Valentin [France] ; Nathan Téné [France] ; Michel Treilhou [France] ; Fakher Chabchoub [Tunisie] ; Françoise Nepveu [France] | New 3-substituted-2,1-benzisoxazoles: Synthesis and antimicrobial activities |
000105 (2017) |
K. Fourmy [France] ; M. Gouygou [France] ; O. Dechy-Cabaret [France] ; F. Benoit-Vical [France] | Gold(I) complexes bearing phosphole ligands: Synthesis and antimalarial activity |
000133 (2015-10-16) |
Chandima S. K. Rajapakse [États-Unis] ; Maryna Lisai [États-Unis] ; Christiane Deregnaucourt [France] ; Véronique Sinou [France] ; Christine Latour [France] ; Dipankar Roy [États-Unis] ; Joseph Schrével [France] ; Roberto A. Sánchez-Delgado [États-Unis] | Synthesis of New 4-Aminoquinolines and Evaluation of Their In Vitro Activity against Chloroquine-Sensitive and Chloroquine-Resistant Plasmodium falciparum |
000134 (2015-10-05) |
Elena Cesar Rodo [France] | Total synthesis of polysubstituted antiparasitic (aza)naphtoquinones |
000153 (2015) |
Chandima S K. Rajapakse [États-Unis] ; Maryna Lisai [États-Unis] ; Christiane Deregnaucourt [France] ; Véronique Sinou [France] ; Christine Latour [France] ; Dipankar Roy [États-Unis] ; Joseph Schrével [France] ; Roberto A. Sánchez-Delgado [États-Unis] | Synthesis of New 4-Aminoquinolines and Evaluation of Their In Vitro Activity against Chloroquine-Sensitive and Chloroquine-Resistant Plasmodium falciparum. |
000171 (2014) |
Nicolas Primas [France] ; Peggy Suzanne [France] ; Pierre Verhaeghe [France] ; Sébastien Hutter [France] ; Charline Kieffer [France] ; Michèle Laget [France] ; Anita Cohen [France] ; Julie Broggi [France] ; Jean-Charles Lancelot [France] ; Aurélien Lesnard [France] ; Patrick Dallemagne [France] ; Pascal Rathelot [France] ; Sylvain Rault [France] ; Patrice Vanelle [France] ; Nadine Azas [France] | Synthesis and in vitro evaluation of 4-trichloromethylpyrrolo[1,2-a]quinoxalines as new antiplasmodial agents |
000213 (2012-04) |
Xiao-Min Yu ; Florence Ramiandrasoa ; Lucie Guetzoyan ; Bruno Pradines ; Edgar Quintino ; Daniele Gadelle ; Patrick Forterre ; Thierry Cresteil [France] ; Jean-Pierre Mahy ; Stéphanie Pethe | Synthesis and biological evaluation of acridine derivatives as antimalarial agents. |
000266 (2009-12-01) |
Lucie Guetzoyan ; Xiao-Min Yu ; Florence Ramiandrasoa ; Stéphanie Pethe ; Christophe Rogier ; Bruno Pradines ; Thierry Cresteil [France] ; Martine Perrée-Fauvet ; Jean-Pierre Mahy | Antimalarial acridines: synthesis, in vitro activity against P. falciparum and interaction with hematin. |
000277 (2009) |
Emilia P Unescu [Roumanie] ; Sophie Susplugas [France] ; Emmanuelle Boll ; Richard Varga [Roumanie] ; Elisabeth Mouray [France] ; Ion Grosu [Roumanie] ; Philippe Grellier [France] ; Patricia Melnyk [France] | Replacement of the 4′‐Hydroxy Group of Amodiaquine and Amopyroquine by Aromatic and Aliphatic Substituents: Synthesis and Antimalarial Activity |
000293 (2008) |
E. Paunescu [France] ; Sophie Susplugas [France] ; E. Boll ; R. Varga ; Elisabeth Mouray [France] ; Philippe Grellier [France] ; Patricia Melnyk [France] | Synthesis and antimalarial activity of new amino analogues of amodiaquine. |
000303 (2008) |
Sandrine Delarue-Cochin [France] ; Philippe Grellier [France] ; Louis Maes [Belgique] ; Elisabeth Mouray [France] ; Christian Sergheraert [France] ; Patricia Melnyk [France] | Synthesis and antimalarial activity of carbamate and amide derivatives of 4-anilinoquinoline |
000307 (2007-06-29) |
Giovanny Garavito [France] | Experimental pharmacological study of the antimalarial activity of a compound of synthesis: the methylthioninium chloride |
000326 (2006) |
Apiwat Baramee [France] ; Alexandra Coppin [France] ; Marlène Mortuaire [France] ; Lydie Pelinski [France] ; Stanislas Tomavo [France] ; Jacques Brocard [France] | Synthesis and in vitro activities of ferrocenic aminohydroxynaphthoquinones against Toxoplasma gondii and Plasmodium falciparum. |
000330 (2006) |
Patricia Melnyk [France] ; Virginie Leroux [France] ; Christian Sergheraert [France] ; Philippe Grellier [France] | Design, synthesis and in vitro antimalarial activity of an acylhydrazone library |
000331 (2006) |
Christophe Biot [France] ; Wassim Daher [France] ; Natascha Chavain [France] ; Thierry Fandeur [France] ; Jamal Khalife [France] ; Daniel Dive [France] ; Erik De Clercq [Belgique] | Design and Synthesis of Hydroxyferroquine Derivatives with Antimalarial and Antiviral Activities |
000340 (2005-02-15) |
Lydie Pélinski [France] ; Dorothée Razafimahefa [Madagascar] ; Marie-Thérèse Martin [France] ; David Ramanitrahasimbola [Madagascar] ; Philippe Rasoanaivo [Madagascar] ; Jacques Brocard [France] | Synthesis and chloroquine-enhancing activity of Na-deacetyl-ferrocenoyl-strychnobrasiline |
000351 (2004-06-14) |
F. Trigalo [France] ; R. Joyeau [France] ; V. C. Pham [France] ; J. J. Youté [France] ; P. Rasoanaivo ; F. Frappier [France] | Synthesis of modulators of chloroquine resistance in Plasmodium falciparum, analogues of malagashanine from strychnobrasiline |