Ident. | Authors (with country if any) | Title |
---|
001849 |
Vivian Cody [États-Unis] ; Jim Pace [États-Unis] ; Sherry F. Queener [États-Unis] ; Ona O. Adair [États-Unis] ; Aleem Gangjee [États-Unis] | Kinetic and Structural Analysis for Potent Antifolate Inhibition of Pneumocystis jirovecii, Pneumocystis carinii, and Human Dihydrofolate Reductases and Their Active-Site Variants |
002E31 |
Aleem Gangjee [États-Unis] ; YING ZHAO [États-Unis] ; Michael A. Innat [États-Unis] ; Jessica E. Thorpe [États-Unis] ; Lora C. Bailey-Downs [États-Unis] ; Roy L. Kisliuk [États-Unis] | Novel tricyclic indeno[2,1-d]pyrimidines with dual antiangiogenic and cytotoxic activities as potent antitumor agents |
002F10 |
Aleem Gangjee [États-Unis] ; Sonali Kurup [États-Unis] ; Michael A. Ihnat [États-Unis] ; Jessica E. Thorpe [États-Unis] ; Bryan Disch [États-Unis] | N4-Aryl-6-substitutedphenylmethyl-7H-pyrrolo[2,3-d]pyrimidine-2,4-diamines as receptor tyrosine kinase inhibitors |
004426 |
XIN ZHANG [États-Unis] ; XILIN ZHOU [États-Unis] ; Roy L. Kisliuk [États-Unis] ; Jennifer Piraino [États-Unis] ; Vivian Cody [États-Unis] ; Aleem Gangjee [États-Unis] | Design, synthesis, biological evaluation and X-ray crystal structure of novel classical 6,5,6-tricyclic benzo[4,5]thieno[2,3-d]pyrimidines as dual thymidylate synthase and dihydrofolate reductase inhibitors |
004566 |
Aleem Gangjee [États-Unis] ; Ojas A. Namjoshi [États-Unis] ; Staci N. Keller [États-Unis] ; Charles D. Smith [États-Unis] | 2-Amino-4-methyl-5-phenylethyl substituted-7-N-benzyl-pyrrolo[2,3-d]pyrimidines as novel antitumor antimitotic agents that also reverse tumor resistance |