Pharmacological potential of Populus nigra extract as antioxidant, anti-inflammatory, cardiovascular and hepatoprotective agent.
Identifieur interne : 002558 ( Main/Exploration ); précédent : 002557; suivant : 002559Pharmacological potential of Populus nigra extract as antioxidant, anti-inflammatory, cardiovascular and hepatoprotective agent.
Auteurs : Nadjet Debbache-Benaida [Algérie] ; Dina Atmani-Kilani ; Valérie Barbara Schini-Keirth ; Nouredine Djebbli ; Djebbar AtmaniSource :
- Asian Pacific journal of tropical biomedicine [ 2221-1691 ] ; 2013.
Descripteurs français
- KwdFr :
- Agents cardiovasculaires (pharmacologie), Agents protecteurs (pharmacologie), Analyse de variance (MeSH), Animaux (MeSH), Anti-inflammatoires (pharmacologie), Carragénane (toxicité), Chlorure d'aluminium (MeSH), Chlorures (toxicité), Composés de l'aluminium (toxicité), Extraits de plantes (composition chimique), Extraits de plantes (pharmacologie), Femelle (MeSH), Flavonoïdes (analyse), Fleurs (composition chimique), Foie (anatomopathologie), Foie (effets des médicaments et des substances chimiques), Lésions hépatiques dues aux substances (anatomopathologie), Lésions hépatiques dues aux substances (traitement médicamenteux), Monoxyde d'azote (métabolisme), Mâle (MeSH), Nitric oxide synthase type III (métabolisme), Oedème (induit chimiquement), Oedème (physiopathologie), Oedème (traitement médicamenteux), Phénols (analyse), Populus (composition chimique), Souris (MeSH), Tanins (analyse).
- MESH :
- analyse : Flavonoïdes, Phénols, Tanins.
- anatomopathologie : Foie, Lésions hépatiques dues aux substances.
- composition chimique : Extraits de plantes, Fleurs, Populus.
- effets des médicaments et des substances chimiques : Foie.
- induit chimiquement : Oedème.
- métabolisme : Monoxyde d'azote, Nitric oxide synthase type III.
- pharmacologie : Agents cardiovasculaires, Agents protecteurs, Anti-inflammatoires, Extraits de plantes.
- physiopathologie : Oedème.
- toxicité : Carragénane, Chlorures, Composés de l'aluminium.
- traitement médicamenteux : Lésions hépatiques dues aux substances, Oedème.
- Analyse de variance, Animaux, Chlorure d'aluminium, Femelle, Mâle, Souris.
English descriptors
- KwdEn :
- Aluminum Chloride (MeSH), Aluminum Compounds (toxicity), Analysis of Variance (MeSH), Animals (MeSH), Anti-Inflammatory Agents (pharmacology), Cardiovascular Agents (pharmacology), Carrageenan (toxicity), Chemical and Drug Induced Liver Injury (drug therapy), Chemical and Drug Induced Liver Injury (pathology), Chlorides (toxicity), Edema (chemically induced), Edema (drug therapy), Edema (physiopathology), Female (MeSH), Flavonoids (analysis), Flowers (chemistry), Liver (drug effects), Liver (pathology), Male (MeSH), Mice (MeSH), Nitric Oxide (metabolism), Nitric Oxide Synthase Type III (metabolism), Phenols (analysis), Plant Extracts (chemistry), Plant Extracts (pharmacology), Populus (chemistry), Protective Agents (pharmacology), Tannins (analysis).
- MESH :
- chemical , analysis : Flavonoids, Phenols, Tannins.
- chemical , chemistry : Plant Extracts.
- chemical , metabolism : Nitric Oxide, Nitric Oxide Synthase Type III.
- chemical , pharmacology : Anti-Inflammatory Agents, Cardiovascular Agents, Plant Extracts, Protective Agents.
- chemical , toxicity : Aluminum Compounds, Carrageenan, Chlorides.
- chemical : Aluminum Chloride.
- chemically induced : Edema.
- chemistry : Flowers, Populus.
- drug effects : Liver.
- drug therapy : Chemical and Drug Induced Liver Injury, Edema.
- pathology : Chemical and Drug Induced Liver Injury, Liver.
- physiopathology : Edema.
- Analysis of Variance, Animals, Female, Male, Mice.
Abstract
OBJECTIVE
To evaluate antioxidant, anti-inflammatory, hepatoprotective and vasorelaxant activities of Populus nigra flower buds ethanolic extract.
METHODS
Antioxidant and anti-inflammatory activities of the extract were assessed using respectively the ABTS test and the animal model of carrageenan-induced paw edema. Protection from hepatic toxicity caused by aluminum was examined by histopathologic analysis of liver sections. Vasorelaxant effect was estimated in endothelium-intact and -rubbed rings of porcine coronary arteries precontracted with high concentration of U46619.
RESULTS
The results showed a moderate antioxidant activity (40%), but potent anti-inflammatory activity (49.9%) on carrageenan-induced mice paw edema, and also as revealed by histopathologic examination, complete protection against AlCl₃-induced hepatic toxicity. Relaxant effects of the same extract on vascular preparation from porcine aorta precontracted with high concentration of U46619 were considerable at 10⁻¹ g/L, and comparable (P>0.05) between endothelium-intact (67.74%, IC₅₀=0.04 mg/mL) and -rubbed (72.72%, IC₅₀=0.075 mg/mL) aortic rings.
CONCLUSIONS
The extract exerted significant anti-inflammatory, hepatoprotective and vasorelaxant activities, the latter being endothelium-independent believed to be mediated mainly by the ability of components present in the extract to exert antioxidant properties, probably related to an inhibition of Ca²⁺ influx.
DOI: 10.1016/S2221-1691(13)60141-0
PubMed: 23998009
PubMed Central: PMC3757277
Affiliations:
Links toward previous steps (curation, corpus...)
Le document en format XML
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<term>Aluminum Compounds (toxicity)</term>
<term>Analysis of Variance (MeSH)</term>
<term>Animals (MeSH)</term>
<term>Anti-Inflammatory Agents (pharmacology)</term>
<term>Cardiovascular Agents (pharmacology)</term>
<term>Carrageenan (toxicity)</term>
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<term>Chlorides (toxicity)</term>
<term>Edema (chemically induced)</term>
<term>Edema (drug therapy)</term>
<term>Edema (physiopathology)</term>
<term>Female (MeSH)</term>
<term>Flavonoids (analysis)</term>
<term>Flowers (chemistry)</term>
<term>Liver (drug effects)</term>
<term>Liver (pathology)</term>
<term>Male (MeSH)</term>
<term>Mice (MeSH)</term>
<term>Nitric Oxide (metabolism)</term>
<term>Nitric Oxide Synthase Type III (metabolism)</term>
<term>Phenols (analysis)</term>
<term>Plant Extracts (chemistry)</term>
<term>Plant Extracts (pharmacology)</term>
<term>Populus (chemistry)</term>
<term>Protective Agents (pharmacology)</term>
<term>Tannins (analysis)</term>
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<term>Agents protecteurs (pharmacologie)</term>
<term>Analyse de variance (MeSH)</term>
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<term>Carragénane (toxicité)</term>
<term>Chlorure d'aluminium (MeSH)</term>
<term>Chlorures (toxicité)</term>
<term>Composés de l'aluminium (toxicité)</term>
<term>Extraits de plantes (composition chimique)</term>
<term>Extraits de plantes (pharmacologie)</term>
<term>Femelle (MeSH)</term>
<term>Flavonoïdes (analyse)</term>
<term>Fleurs (composition chimique)</term>
<term>Foie (anatomopathologie)</term>
<term>Foie (effets des médicaments et des substances chimiques)</term>
<term>Lésions hépatiques dues aux substances (anatomopathologie)</term>
<term>Lésions hépatiques dues aux substances (traitement médicamenteux)</term>
<term>Monoxyde d'azote (métabolisme)</term>
<term>Mâle (MeSH)</term>
<term>Nitric oxide synthase type III (métabolisme)</term>
<term>Oedème (induit chimiquement)</term>
<term>Oedème (physiopathologie)</term>
<term>Oedème (traitement médicamenteux)</term>
<term>Phénols (analyse)</term>
<term>Populus (composition chimique)</term>
<term>Souris (MeSH)</term>
<term>Tanins (analyse)</term>
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<term>Phenols</term>
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<term>Nitric Oxide Synthase Type III</term>
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<keywords scheme="MESH" type="chemical" qualifier="pharmacology" xml:lang="en"><term>Anti-Inflammatory Agents</term>
<term>Cardiovascular Agents</term>
<term>Plant Extracts</term>
<term>Protective Agents</term>
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<keywords scheme="MESH" type="chemical" qualifier="toxicity" xml:lang="en"><term>Aluminum Compounds</term>
<term>Carrageenan</term>
<term>Chlorides</term>
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<term>Phénols</term>
<term>Tanins</term>
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<term>Lésions hépatiques dues aux substances</term>
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<keywords scheme="MESH" qualifier="composition chimique" xml:lang="fr"><term>Extraits de plantes</term>
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<term>Populus</term>
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<term>Edema</term>
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<keywords scheme="MESH" qualifier="effets des médicaments et des substances chimiques" xml:lang="fr"><term>Foie</term>
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<keywords scheme="MESH" qualifier="induit chimiquement" xml:lang="fr"><term>Oedème</term>
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<keywords scheme="MESH" qualifier="métabolisme" xml:lang="fr"><term>Monoxyde d'azote</term>
<term>Nitric oxide synthase type III</term>
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<keywords scheme="MESH" qualifier="pathology" xml:lang="en"><term>Chemical and Drug Induced Liver Injury</term>
<term>Liver</term>
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<keywords scheme="MESH" qualifier="pharmacologie" xml:lang="fr"><term>Agents cardiovasculaires</term>
<term>Agents protecteurs</term>
<term>Anti-inflammatoires</term>
<term>Extraits de plantes</term>
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<keywords scheme="MESH" qualifier="physiopathologie" xml:lang="fr"><term>Oedème</term>
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<keywords scheme="MESH" qualifier="physiopathology" xml:lang="en"><term>Edema</term>
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<term>Chlorures</term>
<term>Composés de l'aluminium</term>
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<keywords scheme="MESH" qualifier="traitement médicamenteux" xml:lang="fr"><term>Lésions hépatiques dues aux substances</term>
<term>Oedème</term>
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<term>Animals</term>
<term>Female</term>
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<term>Mice</term>
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<keywords scheme="MESH" xml:lang="fr"><term>Analyse de variance</term>
<term>Animaux</term>
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<front><div type="abstract" xml:lang="en"><p><b>OBJECTIVE</b>
</p>
<p>To evaluate antioxidant, anti-inflammatory, hepatoprotective and vasorelaxant activities of Populus nigra flower buds ethanolic extract.</p>
</div>
<div type="abstract" xml:lang="en"><p><b>METHODS</b>
</p>
<p>Antioxidant and anti-inflammatory activities of the extract were assessed using respectively the ABTS test and the animal model of carrageenan-induced paw edema. Protection from hepatic toxicity caused by aluminum was examined by histopathologic analysis of liver sections. Vasorelaxant effect was estimated in endothelium-intact and -rubbed rings of porcine coronary arteries precontracted with high concentration of U46619.</p>
</div>
<div type="abstract" xml:lang="en"><p><b>RESULTS</b>
</p>
<p>The results showed a moderate antioxidant activity (40%), but potent anti-inflammatory activity (49.9%) on carrageenan-induced mice paw edema, and also as revealed by histopathologic examination, complete protection against AlCl₃-induced hepatic toxicity. Relaxant effects of the same extract on vascular preparation from porcine aorta precontracted with high concentration of U46619 were considerable at 10⁻¹ g/L, and comparable (P>0.05) between endothelium-intact (67.74%, IC₅₀=0.04 mg/mL) and -rubbed (72.72%, IC₅₀=0.075 mg/mL) aortic rings.</p>
</div>
<div type="abstract" xml:lang="en"><p><b>CONCLUSIONS</b>
</p>
<p>The extract exerted significant anti-inflammatory, hepatoprotective and vasorelaxant activities, the latter being endothelium-independent believed to be mediated mainly by the ability of components present in the extract to exert antioxidant properties, probably related to an inhibition of Ca²⁺ influx.</p>
</div>
</front>
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<Month>05</Month>
<Day>14</Day>
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<Title>Asian Pacific journal of tropical biomedicine</Title>
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<ArticleTitle>Pharmacological potential of Populus nigra extract as antioxidant, anti-inflammatory, cardiovascular and hepatoprotective agent.</ArticleTitle>
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<Abstract><AbstractText Label="OBJECTIVE" NlmCategory="OBJECTIVE">To evaluate antioxidant, anti-inflammatory, hepatoprotective and vasorelaxant activities of Populus nigra flower buds ethanolic extract.</AbstractText>
<AbstractText Label="METHODS" NlmCategory="METHODS">Antioxidant and anti-inflammatory activities of the extract were assessed using respectively the ABTS test and the animal model of carrageenan-induced paw edema. Protection from hepatic toxicity caused by aluminum was examined by histopathologic analysis of liver sections. Vasorelaxant effect was estimated in endothelium-intact and -rubbed rings of porcine coronary arteries precontracted with high concentration of U46619.</AbstractText>
<AbstractText Label="RESULTS" NlmCategory="RESULTS">The results showed a moderate antioxidant activity (40%), but potent anti-inflammatory activity (49.9%) on carrageenan-induced mice paw edema, and also as revealed by histopathologic examination, complete protection against AlCl₃-induced hepatic toxicity. Relaxant effects of the same extract on vascular preparation from porcine aorta precontracted with high concentration of U46619 were considerable at 10⁻¹ g/L, and comparable (P>0.05) between endothelium-intact (67.74%, IC₅₀=0.04 mg/mL) and -rubbed (72.72%, IC₅₀=0.075 mg/mL) aortic rings.</AbstractText>
<AbstractText Label="CONCLUSIONS" NlmCategory="CONCLUSIONS">The extract exerted significant anti-inflammatory, hepatoprotective and vasorelaxant activities, the latter being endothelium-independent believed to be mediated mainly by the ability of components present in the extract to exert antioxidant properties, probably related to an inhibition of Ca²⁺ influx.</AbstractText>
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<ForeName>Nadjet</ForeName>
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<Author ValidYN="Y"><LastName>Schini-Keirth</LastName>
<ForeName>Valérie Barbara</ForeName>
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