Ident. | Authors (with country if any) | Title |
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000022 (2020) |
Yan Li [République populaire de Chine] ; Xingdong Lin [République populaire de Chine] ; Jianqing Hu [République populaire de Chine] ; Jianbo Shuai [République populaire de Chine] ; Yinan Wei [États-Unis] ; Daohang He [République populaire de Chine] | Synthesis and biological evaluation of stilbene-based peptoid mimics against the phytopathogenic bacterium Xanthomonas citri pv. citri. |
000023 (2020) |
Reza Mohammadi [Iran] ; Bahareh Shokri [Iran] ; Danial Shamshirian [Iran] ; Afshin Zarghi [Iran] ; Soraya Shahhosseini [Iran] | Synthesis and biological evaluation of RGD conjugated with Ketoprofen/Naproxen and radiolabeled with [99mTc] via N4(GGAG) for αVβ3 integrin-targeted drug delivery. |
000034 (2020) |
Jing Han [République populaire de Chine] ; Junjie Fu [République populaire de Chine] ; Qimeng Yang [République populaire de Chine] ; Feng Zhou [République populaire de Chine] ; Xinyu Chen [République populaire de Chine] ; Chenglin Li [République populaire de Chine] ; Jian Yin [République populaire de Chine] | Rational design and biological evaluation of gemfibrozil modified Xenopus GLP-1 derivatives as long-acting hypoglycemic agents. |
000046 (2020) |
Jingyi Lu [République populaire de Chine] ; Baijie Ren [République populaire de Chine] ; Lei Wang [République populaire de Chine] ; Minghe Li [République populaire de Chine] ; Yue Liu [République populaire de Chine] | Preparation and Evaluation of IL-1ra-Loaded Dextran/PLGA Microspheres for Inhibiting Periodontal Inflammation In Vitro. |
000067 (2020) |
Safirah Maheen [Pakistan] ; Akhtar Rasul [Pakistan] ; Muhammad Hanif [Pakistan] ; Hafeez Ullah Khan [Pakistan] | Lipospheres for Simultaneous Controlled Release and Improved Pharmacokinetic Profiles of Saxagliptin-Enalapril: Formulation, Optimization, and Comparative In Vitro-In Vivo Evaluation. |
000099 (2020) |
Naik Hardik Jinal [Inde] ; Natarajan Amaresan [Inde] | Evaluation of biocontrol Bacillus species on plant growth promotion and systemic-induced resistant potential against bacterial and fungal wilt-causing pathogens. |
000124 (2020) |
Özge Temiz [Turquie] | Biopesticide emamectin benzoate in the liver of male mice: evaluation of oxidative toxicity with stress protein, DNA oxidation, and apoptosis biomarkers. |
000233 (2019) |
Mohamed Hisham [Égypte] ; Bahaa G M. Youssif [Arabie saoudite] ; Essam Eldin A. Osman [Égypte] ; Alaa M. Hayallah [Égypte] ; Mohamed Abdel-Aziz [Égypte] | Synthesis and biological evaluation of novel xanthine derivatives as potential apoptotic antitumor agents. |
000234 (2019) |
Zhen Guo [République populaire de Chine] ; Xiaowei Song [République populaire de Chine] ; Li-Min Zhao [République populaire de Chine] ; Ming Guan Piao [République populaire de Chine] ; Jishan Quan [République populaire de Chine] ; Hu-Ri Piao [République populaire de Chine] ; Cheng Hua Jin [République populaire de Chine] | Synthesis and biological evaluation of novel benzo[c][1,2,5]thiadiazol-5-yl and thieno[3,2-c]- pyridin-2-yl imidazole derivatives as ALK5 inhibitors. |
000236 (2019) |
Xiaoqing Song [République populaire de Chine] ; Qianqian Gan [République populaire de Chine] ; Xuran Zhang [République populaire de Chine] ; Junbo Zhang [République populaire de Chine] | Synthesis and Biological Evaluation of Novel 99mTc-Labeled Palbociclib Derivatives Targeting Cyclin-Dependent Kinase 4/6 (CDK4/6) as Potential Cancer Imaging Agents. |
000237 (2019) |
Ting Liu [République populaire de Chine] ; Qingxuan Zeng [République populaire de Chine] ; Xiaoqiang Zhao [République populaire de Chine] ; Wei Wei [République populaire de Chine] ; Yinghong Li [République populaire de Chine] ; Hongbin Deng [République populaire de Chine] ; Danqing Song [République populaire de Chine] | Synthesis and Biological Evaluation of Fangchinoline Derivatives as Anti-Inflammatory Agents through Inactivation of Inflammasome. |
000332 (2019) |
Zijian Li [République populaire de Chine] ; Song Zhang [République populaire de Chine] ; Jinxiu Li [République populaire de Chine] ; Huanhuan Zeng [République populaire de Chine] ; Yi Wang [République populaire de Chine] ; Yingru Huang [République populaire de Chine] | Nerve regeneration in rat peripheral nerve allografts: Evaluation of cold-inducible RNA-binding protein in nerve storage and regeneration. |
000383 (2019) |
Mohammed A. Alshehri [Arabie saoudite] ; Piotr M. Wierzbicki [Pologne] ; Hassan F. Kaboo [Égypte] ; Mohamed S M. Nasr [Égypte] ; Mohamed E. Amer [Égypte] ; Tamer M M. Abuamara [Égypte] ; Doaa A. Badr [Égypte] ; Kamel A. Saleh [Arabie saoudite] ; Ahmed E. Fazary [Égypte] ; Aly F. Mohamed [Égypte] | In vitro evaluation of electroporated gold nanoparticles and extremely-low frequency electromagnetic field anticancer activity against Hep-2 laryngeal cancer cells. |
000419 (2019) |
Hui-Yun Zhang [République populaire de Chine] ; Cong-Yong Sun [République populaire de Chine] ; Michael Adu-Frimpong [République populaire de Chine] ; Jiang-Nan Yu [République populaire de Chine] ; Xi-Ming Xu [République populaire de Chine] | Glutathione-sensitive PEGylated curcumin prodrug nanomicelles: Preparation, characterization, cellular uptake and bioavailability evaluation. |
000448 (2019) |
Afsaneh Farjami [Iran] ; Mohammadreza Siahi-Shadbad ; Parvin Akbarzadehlaleh ; Khashayar Roshanzamir ; Ommoleila Molavi | Evaluation of the Physicochemical and Biological Stability of Cetuximab under Various Stress Condition. |
000449 (2019) |
Bruno De Souza Gonçalves [Brésil] ; Jéssica M. De Moura Valadares [Brésil] ; Silmara L G. Alves [Brésil] ; Simone C. Silva [Brésil] ; Luciana P. Rangel [Brésil] ; Vanessa F. Cortes [Brésil] ; José A F P. Villar [Brésil] ; Leandro A. Barbosa [Brésil] ; Hérica De Lima Santos [Brésil] | Evaluation of neuroprotective activity of digoxin and semisynthetic derivatives against partial chemical ischemia. |
000450 (2019) |
Jiake He [République populaire de Chine] ; Ge Zhang [République populaire de Chine] ; Qiuyang Zhang [République populaire de Chine] ; Jiayin Chen [République populaire de Chine] ; Yongjie Zhang [République populaire de Chine] ; Xiaoxia An [République populaire de Chine] ; Pan Wang [République populaire de Chine] ; Shan Xie [République populaire de Chine] ; Fang Fang [République populaire de Chine] ; Jianheng Zheng [République populaire de Chine] ; Yue Tang [République populaire de Chine] ; Jiabi Zhu [République populaire de Chine] ; Yang Yu [République populaire de Chine] ; Xijing Chen [République populaire de Chine] ; Yang Lu [République populaire de Chine] | Evaluation of inhaled recombinant human insulin dry powders: pharmacokinetics, pharmacodynamics and 14-day inhalation. |
000451 (2019) |
Edyta Konecka [Pologne] ; Joanna Mokracka [Pologne] ; Sylwia Krzymi Ska [Pologne] ; Adam Kaznowski [Pologne] | Evaluation of The Pathogenic Potential of Insecticidal Serratia marcescens Strains to Humans. |
000452 (2019) |
Ahmet M. En K [Turquie] ; Çi Dem Çhedef [Turquie] ; Ayfer Y. K Lçar [Turquie] ; Eser Uçar [Turquie] ; Kadir Ar [Turquie] ; Yasemin Parlak [Turquie] ; Elvan S. Bilgin [Turquie] ; Serap Teksöz [Turquie] | Evaluation of New 99mTc(CO)3 + Radiolabeled Glycylglycine In Vivo. |
000453 (2019) |
Caixing Xiong [États-Unis] ; Krzysztof Kaczmarek [Pologne] ; Janusz Zabrocki [Pologne] ; Patricia V. Pietrantonio [États-Unis] ; Ronald J. Nachman [États-Unis] | Evaluation of Aib and PEG-polymer insect kinin analogs on mosquito and tick GPCRs identifies potent new pest management tools with potentially enhanced biostability and bioavailability. |
000487 (2019) |
Fatma A F. Ragab [Égypte] ; Salah A. Abdel-Aziz [Égypte] ; Marwa Kamel [Égypte] ; Abdelsalam Mohamed A. Ouf [Égypte] ; Heba Abdelrasheed Allam [Égypte] | Design, synthesis and biological evaluation of some new 1,3,4-thiadiazine-thiourea derivatives as potential antitumor agents against non-small cell lung cancer cells. |